SCHEMBL27570010

SCHEMBL27570010

CC(C)CCCCCCCCCC(=O)Nc1ncnc2[nH]cnc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DEGS1 O15121 1/20 0.47
XDH P47989 1/20 0.45
PAX8 Q06710 1/20 0.42
HDAC1 Q13547 8/20 0.40
HDAC2 Q92769 6/20 0.40
HDAC3 O15379 5/20 0.36
HDAC6 Q9UBN7 5/20 0.36
HDAC10 Q969S8 3/20 0.36
HDAC8 Q9BY41 3/20 0.36
HDAC9 Q9UKV0 3/20 0.36
HDAC5 Q9UQL6 3/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
ERBB2 P04626 2/20 0.36
KDR P35968 2/20 0.36
BRD4 O60885 4/20 0.35
BRPF1 P55201 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7052321 0.86 XDH (0.61) DEGS1XDHHDAC1HDAC2BRD4
SCHEMBL5193809 0.86 XDH (0.61) DEGS1XDHHDAC1HDAC2BRD4
SCHEMBL2623138 0.85 XDH (0.62) DEGS1XDHHDAC1HDAC2BRD4
SCHEMBL27570011 0.82 HDAC1 (0.58) DEGS1PAX8HDAC1HDAC2BRD4
SCHEMBL1369446 0.82 XDH (0.45) XDHHDAC1HDAC2HDAC3HDAC6
SCHEMBL13538979 0.81 XDH (0.45) XDHHDAC1HDAC2HDAC6HDAC8
Hydrochloric Acid SCHEMBL1370010 0.81 XDH (0.44) XDHHDAC1HDAC2HDAC3NCOR2
SCHEMBL1369225 0.79 XDH (0.41) XDHHDAC1HDAC2BRD4BRPF1
SCHEMBL1371416 0.78 XDH (0.41) XDHHDAC1HDAC2BRD4AURKA
Hydrochloric Acid SCHEMBL1371823 0.78 XDH (0.40) XDHHDAC1HDAC2BRD4BRPF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1343650-A Anticancer compound with particular structure YANG ZHENHUA (CN) 2002-04-10 CN disclosed