SCHEMBL2757571

SCHEMBL2757571

COc1ccccc1CN(C(=O)C[18F])c1cccnc1Oc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TSPO P30536 5/20 0.68
OPRK1 P41145 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2757569 0.93 TSPO (0.58) TSPO
SCHEMBL2757570 0.90 TSPO (0.69) TSPOOPRK1
SCHEMBL242089 0.88 TSPO (0.67) TSPO
SCHEMBL12374085 0.84 TSPO (0.52) TSPOOPRK1
SCHEMBL2757568 0.83 MAPK8 (0.47) TSPO
SCHEMBL13492581 0.82 TSPO (0.47) TSPOOPRK1
SCHEMBL3268801 0.82 TSPO (0.45) TSPOOPRK1
SCHEMBL13161737 0.81 TSPO (0.57) TSPOOPRK1
SCHEMBL241634 0.80 TSPO (0.62) TSPOOPRK1
SCHEMBL2757555 0.80 TSPO (0.62) TSPOOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120003154-A1 ARYLOXYANILIDE DERIVATIVES GE HEALTHCARE LIMITED (GB) 2012-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120003154-A1 ARYLOXYANILIDE DERIVATIVES GABBR1, GABRA4, CNR1 TSPO 43/4885OPRK1 57/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.