SCHEMBL27577249

SCHEMBL27577249

O=C(NC(Cc1c[nH]c2ccccc12)c1nc(-c2ccccc2)c[nH]1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.54
CYP3A4 P08684 1/20 0.53
CYP2C19 P33261 1/20 0.53
TACR1 P25103 9/20 0.52
ITGB2 P05107 1/20 0.51
ICAM1 P05362 1/20 0.51
ITGAL P20701 1/20 0.51
SSTR3 P32745 2/20 0.50
ERAP2 Q6P179 1/20 0.50
SSTR1 P30872 1/20 0.49
HPGDS O60760 1/20 0.48
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1927953 1.00 CTSL (0.54) CTSLCYP3A4CYP2C19TACR1ITGB2
SCHEMBL2342532 0.90 SSTR3 (0.52) ITGB2ICAM1ITGALSSTR3SSTR1
SCHEMBL1928434 0.88 SSTR3 (0.46) CTSLTACR1ITGB2ICAM1ITGAL
SCHEMBL4244384 0.86 KMT2A (0.59) SSTR3SSTR1MEN1KMT2A
SCHEMBL1927088 0.86 FPR2 (0.56) ITGB2ICAM1ITGALSSTR3SSTR1
SCHEMBL27564526 0.86 FPR2 (0.56) ITGB2ICAM1ITGALSSTR3SSTR1
SCHEMBL13579138 0.85 SSTR3 (0.49) TACR1ITGB2ICAM1ITGALSSTR3
SCHEMBL4247165 0.85 KMT2A (0.54) SSTR3SSTR1KMT2A
SCHEMBL1723433 0.84 SSTR3 (0.47) ITGB2ICAM1ITGALSSTR3SSTR1
SCHEMBL14341130 0.84 SSTR3 (0.48) TACR1ITGB2ICAM1ITGALSSTR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1391474-A 5-membered heterocyclic derivatives, their preparation and their use as medicaments SOD CONSEILS RECH APPLIC (FR) 2003-01-15 CN claimed