Methane

Methane

SCHEMBL27587790

C.N#Cc1cc(Br)c2ncccc2c1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.41
GLO1 Q04760 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SLC40A1 Q9NP59 2/20 0.40
TTR P02766 1/20 0.40
ALB P02768 1/20 0.40
CCR1 P32246 3/20 0.39
CCR8 P51685 3/20 0.39
HTT P42858 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
HSP90AA1 P07900 1/20 0.39
MMP2 P08253 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
MMP9 P14780 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3925761 0.78 CCR1 (0.50) HPGDSGLO1SLC40A1CCR1CCR8
SCHEMBL20306596 0.78 PKM (0.49) HPGDSGLO1MEN1KMT2ASLC40A1
SCHEMBL1994732 0.75 CCR1 (0.57) HPGDSGLO1MEN1KMT2ASLC40A1
SCHEMBL30492680 0.75 CCR1 (0.57) HPGDSGLO1MEN1KMT2ASLC40A1
SCHEMBL662676 0.74 KDM4E (0.47) MEN1KMT2ACCR1CCR8HTT
SCHEMBL2582442 0.73 CCR1 (0.46) MEN1KMT2ASLC40A1CCR1CCR8
SCHEMBL31276857 0.73 CCR1 (0.46) MEN1KMT2ASLC40A1CCR1CCR8
SCHEMBL4025285 0.72 PDE4A (0.39) MEN1KMT2ACCR1CCR8HTT
Water SCHEMBL28285432 0.72 LMNA (0.61) MEN1KMT2ACCR1CCR8HTT
SCHEMBL15007502 0.72 KDM4E (0.48) MEN1KMT2ACCR1CCR8HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100508978-C Substituted 8-arylquinoline phosphodiesterase-4 inhibitors MERCK & CO INC MERCK FROSST CA (US) 2009-07-08 CN disclosed
CN-1551769-A Substituted 8-arylquinoline phosphodiesterase-4 inhibitors 2004-12-01 CN disclosed