SCHEMBL27588293

SCHEMBL27588293

C=CCOC(=O)c1ccccc1NC(=O)OC(C)(C)C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.57
ALDH1A1 P00352 6/20 0.51
HSD17B10 Q99714 4/20 0.51
TSHR P16473 3/20 0.51
RXFP1 Q9HBX9 1/20 0.49
LMNA P02545 5/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 6/20 0.43
HTT P42858 2/20 0.41
IDO1 P14902 1/20 0.41
USP2 O75604 1/20 0.41
HPGD P15428 1/20 0.41
TP53 P04637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28493853 0.84 KDM4E (0.60) ALDH1A1HSD17B10TSHRLMNACYP1A2
SCHEMBL29663621 0.82 RXFP1 (0.55) ALDH1A1HSD17B10TSHRRXFP1LMNA
SCHEMBL12872990 0.82 ALDH1A1 (0.56) CYP3A4ALDH1A1TSHRRXFP1LMNA
SCHEMBL9330701 0.81 KMT2A (0.61) ALDH1A1HSD17B10TSHRRXFP1LMNA
SCHEMBL7600019 0.80 CYP3A4 (0.55) CYP3A4ALDH1A1HSD17B10TSHRLMNA
SCHEMBL13209432 0.80 RXFP1 (0.46) ALDH1A1RXFP1LMNACYP1A2CYP2C19
SCHEMBL12292165 0.79 RXFP1 (0.53) ALDH1A1HSD17B10TSHRRXFP1LMNA
SCHEMBL2460812 0.79 CYP3A4 (0.70) CYP3A4ALDH1A1HSD17B10TSHRLMNA
SCHEMBL11302755 0.79 CYP3A4 (0.60) CYP3A4ALDH1A1HSD17B10TSHRLMNA
SCHEMBL7581997 0.79 CYP3A4 (0.60) CYP3A4ALDH1A1HSD17B10TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100413972-C Enzymatic process for preparing substituted 2-amino-3- (2-amino-thiophenyl) -propionic acids HOFFMANN LA ROCHE (CH) 2008-08-27 CN disclosed
CN-1553959-A Enzymatic process for preparing substituted 2-amino-3- (2-amino-thiophenyl) -propionic acids - 2004-12-08 CN disclosed