SCHEMBL9330701

SCHEMBL9330701

COC(=O)c1ccccc1NC(=O)OC(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.61
KDM4E B2RXH2 6/20 0.57
ALDH1A1 P00352 6/20 0.57
HPGD P15428 4/20 0.57
CYP1A2 P05177 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
CYP2C19 P33261 2/20 0.57
POLB P06746 1/20 0.57
ATM Q13315 1/20 0.57
HSD17B10 Q99714 5/20 0.55
TSHR P16473 3/20 0.55
GAA P10253 2/20 0.55
MAPT P10636 2/20 0.55
MAPK1 P28482 1/20 0.55
RXFP1 Q9HBX9 1/20 0.54
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
ALOX15 P16050 1/20 0.53
CYP2D6 P10635 1/20 0.52
ALOX12 P18054 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29663621 0.92 RXFP1 (0.55) KMT2AKDM4EALDH1A1HPGDCYP1A2
SCHEMBL12292165 0.89 RXFP1 (0.53) KMT2AKDM4EALDH1A1HPGDCYP1A2
SCHEMBL28033115 0.88 RXFP1 (0.52) KMT2AKDM4EALDH1A1HPGDCYP1A2
SCHEMBL28476853 0.86 KDM4E (0.51) KMT2AKDM4EALDH1A1HPGDCYP1A2
SCHEMBL15440466 0.86 RXFP1 (0.48) KMT2AKDM4EALDH1A1HPGDCYP1A2
SCHEMBL29992092 0.85 RXFP1 (0.59) KMT2ACYP2C19POLBRXFP1LMNA
SCHEMBL29702265 0.85 RXFP1 (0.55) KMT2AKDM4ESMN1; SMN2POLBRXFP1
SCHEMBL15368377 0.85 RXFP1 (0.59) KMT2ACYP2C19POLBRXFP1LMNA
SCHEMBL222446 0.85 RXFP1 (0.55) KMT2AKDM4ESMN1; SMN2POLBRXFP1
SCHEMBL3771942 0.85 RXFP1 (0.50) KMT2AKDM4EALDH1A1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073741-B Phthalazinones and isoquinolinones as ROCK inhibitors 百时美施贵宝公司 2017-08-08 CN disclosed
CN-103992326-A Indol-hexahydropyrazine-quinazolinone anti-tumour compounds and preparation method thereof UNIV PLA 2ND MILITARY MEDICAL 2014-08-20 CN disclosed
CN-1653042-A Aminoalcohol derivatives as beta-3 adrenergic receptor agonists FUJISAWA PHARMACEUTICAL CO (JP) 2005-08-10 CN disclosed
US-5298409-A Of esters, antigen diastereomers which are stable analogs of the unstable ester transition states THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-03-29 US disclosed
US-5190865-A Antibody-enhanced stereospecific hydrolyses THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1993-03-02 US disclosed