SCHEMBL27591986

SCHEMBL27591986

CCCCCCNc1nc(N)nc(-c2ccccc2)c1C#N

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 3/20 0.58
ADORA1 P30542 16/20 0.56
ADORA2A P29274 15/20 0.56
ADORA2B P29275 3/20 0.49
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
CYP2C19 P33261 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441739 0.90 ADORA1 (0.61) TLR8ADORA1ADORA2AADORA2B
SCHEMBL6443635 0.84 ADORA1 (0.57) TLR8ADORA1ADORA2AADORA2BKDM4E
SCHEMBL6443028 0.81 ADORA1 (0.60) ADORA1ADORA2AADORA2BKDM4EALDH1A1
SCHEMBL28748293 0.80 ADORA1 (0.56) TLR8ADORA1ADORA2AADORA2B
SCHEMBL6443545 0.79 ADORA1 (0.63) ADORA1ADORA2AADORA2B
SCHEMBL6443531 0.77 ADORA2A (0.55) TLR8ADORA1ADORA2AADORA2BKDM4E
SCHEMBL6442358 0.77 ADORA1 (0.63) ADORA1ADORA2AADORA2BKDM4EALDH1A1
SCHEMBL20434287 0.76 TLR8 (0.66) TLR8
SCHEMBL6445232 0.74 ACHE (0.56) ADORA1ADORA2AKDM4EALDH1A1LMNA
SCHEMBL6440910 0.74 ADORA1 (1.00) ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1438890-A Adenosine receptor modulators HOFFMANNLA ROCHE AG F (CH) 2003-08-27 CN disclosed