SCHEMBL27592575

SCHEMBL27592575

CC(C)(C)c1ccnc(N)c1C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 9/20 0.40
NOS3 P29474 8/20 0.40
NOS1 P29475 5/20 0.35
PRKCI P41743 1/20 0.33
F12 P00748 1/20 0.33
PLAU P00749 1/20 0.33
NCF1 P14598 1/20 0.33
BACE1 P56817 1/20 0.33
ALOX5AP P20292 5/20 0.33
FEN1 P39748 5/20 0.33
NUDT1 P36639 2/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL984332 0.80 NOS2 (0.52) NOS2NOS3NOS1PRKCIF12
SCHEMBL4539853 0.78 NOS2 (0.56) NOS2NOS3NOS1PRKCIF12
SCHEMBL16414488 0.78 CXCR4 (0.32)
SCHEMBL15889710 0.77 NOS2 (0.39) NOS2NOS3NOS1PRKCIF12
SCHEMBL20989742 0.77 NOS2 (0.39) NOS2NOS3NOS1PRKCIF12
SCHEMBL31050050 0.77 NOS2 (0.39) NOS2NOS3NOS1PRKCIF12
SCHEMBL18590248 0.77 ALOX5AP (0.39) NOS2NOS3NOS1PRKCIF12
SCHEMBL30465794 0.76 CYP2A6 (0.34)
SCHEMBL3635124 0.76 CYP3A4 (0.30)
SCHEMBL2029268 0.76 CYP2A6 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100338088-C 2-substituted pregna-1,3,5(10)-triene and chola-1,3,5(10)-triene derivatives and their biological activity RES INST MEDICINE CHEM (US) 2007-09-19 CN disclosed
CN-1444597-A 2-substituted pregna-1, 3,5(10) -triene and chol-1, 3,5(10) -triene derivatives and their biological activity RES INST MEDICINE CHEM (US) 2003-09-24 CN disclosed