SCHEMBL27596181

SCHEMBL27596181

Cc1ccccc1C(=O)c1cnc(NC(C)CCOS(=O)(=O)c2cccs2)s1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.36
MAPK13 O15264 4/20 0.35
MAPK12 P53778 4/20 0.35
MAPK11 Q15759 4/20 0.35
ALDH1A1 P00352 1/20 0.35
LCK P06239 2/20 0.35
CTNNB1 P35222 1/20 0.34
WNT3A P56704 1/20 0.34
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27596141 0.87 MAPK14 (0.39) MAPK14MAPK13MAPK12MAPK11
SCHEMBL27614917 0.85 F2 (0.37) MAPK14MAPK13MAPK12MAPK11ALDH1A1
SCHEMBL27596187 0.77 MAPK14 (0.45) MAPK14MAPK13MAPK12MAPK11LCK
SCHEMBL5564692 0.77 MAPK14 (0.45) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL27614922 0.74 MAPK13 (0.48) MAPK14MAPK13MAPK12MAPK11
SCHEMBL5568018 0.73 NPY5R (0.48) CYP2C9CYP2C19
SCHEMBL5564465 0.73 NPY5R (0.51) CYP2C9CYP2C19
SCHEMBL4429774 0.73 CCR8 (0.35) MAPK14MAPK13MAPK12MAPK11LCK
SCHEMBL27614995 0.72 MAPK14 (0.40) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL5564038 0.71 MAPT (0.43) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100363362-C Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2008-01-23 CN claimed
CN-1639158-A Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2005-07-13 CN claimed
CN-100363362-C Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2008-01-23 CN disclosed
CN-1639158-A Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2005-07-13 CN disclosed