SCHEMBL27607993

SCHEMBL27607993

Nc1cc(CCC(=O)O)cc(-c2ccc3[nH]ncc3c2)c1OCCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.43
ROCK2 O75116 8/20 0.42
ROCK1 Q13464 7/20 0.42
FFAR1 O14842 1/20 0.41
GSK3B P49841 4/20 0.41
CDK5 Q00535 4/20 0.41
DYRK1A Q13627 4/20 0.41
CLK2 P49760 3/20 0.41
CLK4 Q9HAZ1 3/20 0.41
DYRK3 O43781 2/20 0.41
CLK1 P49759 1/20 0.41
CLK3 P49761 1/20 0.41
CDK5R1 Q15078 1/20 0.41
DYRK2 Q92630 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
ATR Q13535 1/20 0.41
CTNNB1 P35222 1/20 0.40
WNT3A P56704 1/20 0.40
AURKB Q96GD4 4/20 0.40
CDC7 O00311 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3882436 0.89 TRPA1 (0.45) TRPA1ROCK2FFAR1GSK3BCDK5
SCHEMBL3882985 0.85 CTNNB1 (0.43) TRPA1ROCK2FFAR1GSK3BCTNNB1
SCHEMBL28752889 0.85 FFAR4 (0.44) FFAR1CTNNB1WNT3A
SCHEMBL27627114 0.85 FFAR1 (0.46) TRPA1ROCK2ROCK1FFAR1GSK3B
SCHEMBL27627100 0.84 FFAR1 (0.51) FFAR1
SCHEMBL923645 0.83 TRPA1 (0.41) TRPA1ROCK2ROCK1GSK3BCDK5
SCHEMBL3882299 0.83 FFAR1 (0.43) TRPA1ROCK2ROCK1FFAR1GSK3B
SCHEMBL3676420 0.81 THRA (0.47) TRPA1ROCK2ROCK1FFAR1GSK3B
SCHEMBL3880425 0.81 TRPA1 (0.47) TRPA1ROCK2FFAR1GSK3BCDK5
SCHEMBL922973 0.81 CDC7 (0.40) TRPA1ROCK2FFAR1ATRCDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100387576-C Substituted phenylalkanoic acid derivatives and use thereof ASAHI CHEMICAL IND (JP) 2008-05-14 CN claimed
CN-1653032-A Substituted phenylalkanoic acid derivatives and use thereof ASAHI CHEMICAL IND (JP) 2005-08-10 CN claimed
CN-100387576-C Substituted phenylalkanoic acid derivatives and use thereof ASAHI CHEMICAL IND (JP) 2008-05-14 CN disclosed
CN-1653032-A Substituted phenylalkanoic acid derivatives and use thereof ASAHI CHEMICAL IND (JP) 2005-08-10 CN disclosed