SCHEMBL27612450

SCHEMBL27612450

Oc1cccc(-c2ncc(-c3ccccc3)cn2)c1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.63
RAB9A P51151 3/20 0.63
NFKB1 P19838 2/20 0.63
NFKB2 Q00653 2/20 0.63
RELA Q04206 2/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
HSD17B1 P14061 9/20 0.59
HSD17B2 P37059 9/20 0.59
CYP3A4 P08684 2/20 0.54
CYP2C9 P11712 2/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
ADORA1 P30542 1/20 0.47
METAP2 P50579 1/20 0.47
KDM4E B2RXH2 1/20 0.46
FYN P06241 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21313422 0.86 NPC1 (0.65) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL3226145 0.81 CHEK1 (0.55) HSD17B1HSD17B2CYP3A4CYP2C9METAP2
SCHEMBL21944933 0.81 HSD17B1 (0.59) HSD17B1HSD17B2CYP3A4CYP2C9METAP2
SCHEMBL28489934 0.80 MEN1 (0.83) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL27625438 0.79 HSD17B1 (0.68) HSD17B1HSD17B2CYP3A4CYP2C9METAP2
SCHEMBL26503498 0.79 NPC1 (0.81) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL2117282 0.79 NPC1 (1.00) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL51869 0.79 HSD17B1 (0.84) HSD17B1HSD17B2CYP3A4CYP2C9MEN1
SCHEMBL29356013 0.79 HSD17B1 (0.84) HSD17B1HSD17B2CYP3A4CYP2C9MEN1
SCHEMBL27960514 0.78 HSD17B1 (0.65) SMN1; SMN2HSD17B1HSD17B2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1678321-A Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds RIGEL PHARMACEUTICALS INC (US) 2005-10-05 CN disclosed