SCHEMBL27615795

SCHEMBL27615795

CC(C)N1CCN(C(=O)c2ccc(CC3CCNCC3)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 11/20 0.59
KCNH2 Q12809 1/20 0.56
CHRNA7 P36544 1/20 0.50
CHRM2 P08172 2/20 0.45
GAA P10253 1/20 0.45
HTT P42858 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
EPHX2 P34913 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27569299 0.84 L3MBTL3 (0.56) GAAHTTCA12CA1CA2
SCHEMBL27634694 0.84 TPSAB1 (0.48) HRH3KCNH2CHRM2
Hydrochloric Acid SCHEMBL4794010 0.83 L3MBTL3 (0.54) GAAHTTCA12CA1CA2
Hydrochloric Acid SCHEMBL4772777 0.80 GAA (0.61) HRH3GAAHTTCA12CA1
SCHEMBL3916721 0.77 HRH3 (0.72) HRH3CHRNA7EPHX2
SCHEMBL12736124 0.77 TPSAB1 (0.53) HRH3KCNH2
SCHEMBL4773726 0.76 GBA1 (0.51)
SCHEMBL1177694 0.75 HRH3 (0.89) HRH3CHRNA7
SCHEMBL20245324 0.75 HRH3 (0.69) HRH3CHRNA7EPHX2
SCHEMBL4237305 0.75 HRH3 (0.61) HRH3KCNH2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100558718-C Piperazinyl and diazacyclo heptyl benzene methane amide and thiobenzamide JANSSEN PHARMACEUTICA NV (BE) 2009-11-11 CN disclosed
CN-1729180-A Piperazinyl and diazapanyl benzamides and benzthioamides JANSSEN PHARMACEUTICA NV (BE) 2006-02-01 CN disclosed