SCHEMBL27616615

SCHEMBL27616615

O=C(O)C(=O)c1cn(C2CCN(Cc3ccccc3)CC2)c2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.60
PRKCG P05129 2/20 0.53
PRKCB P05771 2/20 0.53
PRKCA P17252 2/20 0.53
PRKCH P24723 2/20 0.53
PRKCE Q02156 2/20 0.53
PRKCD Q05655 2/20 0.53
CAMK2D Q13557 2/20 0.53
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
DRD4 P21917 6/20 0.48
DRD2 P14416 5/20 0.48
DRD3 P35462 5/20 0.48
NPSR1 Q6W5P4 1/20 0.47
KDM4E B2RXH2 1/20 0.47
CAMK2B Q13554 1/20 0.47
CAMK2G Q13555 1/20 0.47
CAMK2A Q9UQM7 1/20 0.47
ADORA1 P30542 1/20 0.46
SERPINE1 P05121 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4989734 0.88 HTR6 (0.55) HTR6PRKCGPRKCBPRKCAPRKCH
SCHEMBL4990643 0.79 HTR6 (0.58) HTR6PRKCGPRKCBPRKCAPRKCH
SCHEMBL4988531 0.77 HTR6 (0.56) HTR6PRKCGPRKCBPRKCAPRKCH
SCHEMBL13915330 0.77 PRKCG (0.55) HTR6PRKCGPRKCBPRKCAPRKCH
SCHEMBL4074930 0.75 HTR6 (1.00) HTR6PRKCGPRKCBPRKCAPRKCH
SCHEMBL5625905 0.74 ADORA1 (0.78) NPSR1KDM4EADORA1SERPINE1
SCHEMBL12486470 0.73 KDM4E (0.69) HTR6NPSR1KDM4E
SCHEMBL588318 0.73 PRKCG (0.55) PRKCGPRKCBPRKCAPRKCHPRKCE
SCHEMBL11770132 0.72 KDM4E (0.64) NPSR1KDM4E
SCHEMBL15856599 0.71 KDM4E (0.56) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1639152-A Pyrrole-2, 5-dione derivatives and their use as GSK-3 inhibitors LILLY CO ELI (US) 2005-07-13 CN disclosed