SCHEMBL27623946

SCHEMBL27623946

O=C(c1cccc(-c2ccncc2)c1)c1cccc(-c2ccncc2)c1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
AURKA O14965 3/20 0.52
KMO O15229 2/20 0.52
PRKCI P41743 1/20 0.52
MAPK14 Q16539 2/20 0.51
ATM Q13315 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
NOTUM Q6P988 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.48
HDAC8 Q9BY41 1/20 0.47
KIF11 P52732 1/20 0.47
CNR1 P21554 1/20 0.46
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL207161 0.86 KMO (0.71) AURKAKMOPRKCINOTUMHDAC8
SCHEMBL29627221 0.86 KMO (0.71) AURKAKMOPRKCINOTUMHDAC8
SCHEMBL17742693 0.85 FYN (0.56) AURKAKMOPRKCIKIF11
SCHEMBL31532683 0.85 FYN (0.56) AURKAKMOPRKCIKIF11
SCHEMBL30860478 0.85 FYN (0.57) AURKAKMOPRKCI
SCHEMBL207988 0.85 AURKA (0.50) AURKAKMOPRKCINOTUMSIRT2
SCHEMBL1382873 0.85 FYN (0.57) AURKAKMOPRKCI
SCHEMBL16108896 0.83 KMO (0.56) MEN1KMT2AAURKAKMOPRKCI
Hydrochloric Acid SCHEMBL30037727 0.83 FYN (0.56) AURKAKMOPRKCI
SCHEMBL16858233 0.83 KMO (0.72) MEN1KMT2AKMOATMTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN claimed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN claimed
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN disclosed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN disclosed