SCHEMBL207988

SCHEMBL207988

O=C(Cl)c1cccc(-c2ccncc2)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AURKA O14965 4/20 0.50
KMO O15229 2/20 0.49
PRKCI P41743 1/20 0.49
CNR1 P21554 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.46
NOTUM Q6P988 1/20 0.45
HDAC8 Q9BY41 1/20 0.44
KIF11 P52732 1/20 0.44
HDAC2 Q92769 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
P4HB P07237 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28032601 0.88 KMO (0.59) KMOHDAC8RXRARXRBALDH1A1
SCHEMBL726087 0.86 KMO (0.56) KMOHDAC8RXRARXRBALDH1A1
SCHEMBL27623946 0.85 MEN1 (0.55) AURKAKMOPRKCICNR1SIRT2
SCHEMBL699008 0.84 KMO (0.67) KMOHDAC8RXRARXRBALDH1A1
SCHEMBL30698052 0.84 KMO (0.67) KMOHDAC8RXRARXRBALDH1A1
SCHEMBL207161 0.83 KMO (0.71) AURKAKMOPRKCINOTUMHDAC8
SCHEMBL29627221 0.83 KMO (0.71) AURKAKMOPRKCINOTUMHDAC8
Hydrogen Sulfide SCHEMBL27896825 0.82 KMO (0.64) KMOHDAC8RXRARXRBALDH1A1
SCHEMBL726544 0.82 KMO (0.53) KMOHDAC8RXRARXRBALDH1A1
SCHEMBL205967 0.82 KMO (0.73) KMOCNR1SIRT2ALDH1A1P4HB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108299478-B Cadmium-based metal organic framework material and preparation method and application thereof 华南师范大学 2020-03-24 CN claimed
CN-109627450-B 3D lanthanide metal coordination polymer and synthesis method and application thereof 华南师范大学 2021-03-02 CN disclosed
CN-108299478-B Cadmium-based metal organic framework material and preparation method and application thereof 华南师范大学 2020-03-24 CN disclosed
US-8088760-B2 Benzoxazole carboxamide inhibitors of poly(ADP-ribose)polymerase (PARP) BIOMARIN PHARMACEUTICAL INC. (US) 2012-01-03 US disclosed
EP-2247600-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Lead Therapeutics, Inc. (US) 2010-11-10 EP disclosed
WO-2009099736-A2 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-13 WO disclosed
US-20090197863-A1 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) LEAD THERAPEUTICS, INC. (US) 2009-08-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090197863-A1 BENZOXAZOLE CARBOXAMIDE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) PARP1, PARP2, PARP11 AURKA 2074/4885KMO 985/4885PRKCI 989/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.