SCHEMBL27623968

SCHEMBL27623968

O=C(c1ccc(-c2cccs2)o1)c1ccc(-c2cccs2)o1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 2/20 0.58
ALDH1A1 P00352 5/20 0.54
HPGD P15428 4/20 0.54
KDM4E B2RXH2 3/20 0.54
MAPT P10636 3/20 0.54
HSD17B10 Q99714 2/20 0.54
CACNA1B Q00975 1/20 0.54
APBA1 Q02410 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
PTPRS Q13332 1/20 0.43
SMN1; SMN2 Q16637 6/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
LMNA P02545 4/20 0.41
ESR1 P03372 1/20 0.41
RAB9A P51151 7/20 0.41
NPC1 O15118 6/20 0.41
TP53 P04637 3/20 0.41
GAA P10253 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL375593 0.87 S1PR4 (0.57) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL28750265 0.86 S1PR4 (0.56) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL375486 0.83 S1PR4 (0.60) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL499141 0.80 ALDH1A1 (0.53) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL10252888 0.73 NPC1 (0.64) S1PR4ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL18169219 0.73 ALDH1A1 (0.73) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL5605299 0.71 HPGD (0.48) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL4700249 0.71 CHRNA7 (0.53) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL18876413 0.71 ALDH1A1 (0.46) S1PR4ALDH1A1HPGDKDM4EMAPT
SCHEMBL3348926 0.71 S1PR4 (0.48) S1PR4ALDH1A1HPGDKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN claimed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN claimed
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN disclosed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN disclosed