SCHEMBL27628702

SCHEMBL27628702

CC(C)(C)C(=O)ON1CCC(NC(=O)c2cc(F)cnc2Cl)CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 2/20 0.46
MCHR1 Q99705 1/20 0.41
OPRK1 P41145 1/20 0.40
HPGD P15428 2/20 0.39
SMO Q99835 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4D Q08499 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
DRD3 P35462 2/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
CRHR1 P34998 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5768960 0.84 TP53 (0.51) LMNATP53
SCHEMBL4191215 0.81 HPGD (0.44) SSTR4HPGDPDE4APDE4BPDE4D
SCHEMBL8353152 0.81 HPGD (0.44) SSTR4HPGDPDE4APDE4BPDE4D
SCHEMBL5840688 0.81 HPGD (0.44) SSTR4HPGDPDE4APDE4BPDE4D
SCHEMBL5747378 0.81 HPGDS (0.45) SSTR4MCHR1OPRK1HPGDPDE4B
SCHEMBL8352231 0.78 HPGD (0.50) MCHR1HPGDPDE4APDE4BPDE4D
SCHEMBL27609552 0.78 NPC1 (0.46) OPRK1HPGDLMNA
SCHEMBL3174715 0.78 NPC1 (0.58) OPRK1HPGDLMNA
SCHEMBL8353042 0.77 HPGD (0.51) MCHR1HPGDPDE4APDE4BPDE4D
SCHEMBL5778940 0.77 HPGD (0.51) HPGDPDE4APDE4BPDE4DIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1652782-A Nicotinamide derivatives useful as PDE4 inhibitors PFIZER (US) 2005-08-10 CN disclosed