Rivastigmine

Rivastigmine

SCHEMBL2763

CCN(C)C(=O)Oc1cccc([C@H](C)N(C)C)c1.O=C(O)C(O)C(O)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBCHE

The experimentally established mechanism targets of Rivastigmine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 16/20 1.00
BCHE known ✓ P06276 11/20 1.00
MARK4 Q96L34 1/20 1.00
FAAH O00519 1/20 0.86
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rivastigmine SCHEMBL25232361 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL29779663 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL3978590 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL29612619 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL30064255 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL13841811 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL29614698 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL1170429 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL6382107 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL6382629 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9583 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250382291-A1 SUBSTITUTED PYRROLO[2,3-b]PYRIDINES FOR SUPPRESSING TOXIC ENDOPLASMIC RETICULUM STRESS UNIV COLUMBIA (US) 2025-12-18 US claimed
US-20250333435-A1 TIMOSAPONIN COMPOUNDS GOLDPORP PHARMA LTD (CN) 2025-10-30 US claimed
US-20250329454-A1 DIAGNOSTIC INDICES FOR NEURODEGENERATIVE CONDITIONS CHASE THERAPEUTICS CORP (US) 2025-10-23 US claimed
US-20250304565-A1 NOVEL BENZOFURAN, BENZOTHIOPHENE, AND INDOLE ANALOGS THAT INHIBIT THE FORMATION OF TAU OLIGOMERS AND THEIR METHOD OF USE Oligomerix Inc. (US) 2025-10-02 US claimed
EP-3562483-B1 NOVEL BENZOFURAN, BENZOTHIOPHENE, AND INDOLE ANALOGS THAT INHIBIT THE FORMATION OF TAU OLIGOMERS AND THEIR METHOD OF USE OLIGOMERIX INC (US) 2025-09-03 EP claimed
US-20250214984-A1 COMPOUND HAVING KDM5 INHIBITORY ACTIVITY AND PHARMACEUTICAL USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2025-07-03 US claimed
EP-4146645-B1 3-AZABICYCLO(3.1.0)HEXANE DERIVATIVES HAVING KDM5 INHIBITORY ACTIVITY AND USE THEREOF ONO PHARMACEUTICAL CO (JP) 2025-06-25 EP claimed
US-20250134959-A1 GRANULOCYTE-MACROPHAGE COLONY-STIMULATING FACTOR-BASED TREATMENTS FOR NEURODEGENERATIVE OR NEUROLOGICAL DISEASES OR DISORDERS PARTNER THERAPEUTICS, INC. 2025-05-01 US claimed
CN-119896733-A Compound, preparation method and medical application thereof 百泰生物药业有限公司 2025-04-29 CN claimed
CN-119790152-A Treatment of neurological disorders using modulators of UNC13A gene transcripts 奎里斯公司 2025-04-08 CN claimed
WO-2003041563-A2 NEUROTRANSMITTER BALANCE CHEMOTHERAPY BE ABLE, LLC (US) 2003-05-22 WO claimed
EP-1311511-A1 PYRAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS FOR MODULATING OR INHIBITING ERAB OR HADH2 ACTIVITY Agouron Pharmaceuticals, Inc. (US) 2003-05-21 EP claimed
US-20020151591-A1 Combination use of acetylcholinesterase inhibitors and GABAa inverse agonists for the treatment of cognitive disorders NEUROGEN CORPORATION 2002-10-17 US claimed
US-20020091145-A1 Behavior chemotherapy EIG MARK H (US) 2002-07-11 US claimed
US-20020065292-A1 For use in therapy of neurodegenerative diseases and certain cancers AGOURON PHARMACEUTICALS, INC. 2002-05-30 US claimed
WO-2002032412-A2 COMBINATION USE OF ACETYLCHOLINESTERASE INHIBITORS AND GABAA INVERSE AGONISTS FOR THE TREATMENT OF COGNITIVE DISORDERS PFIZER PRODUCTS INC. (US) 2002-04-25 WO claimed
WO-2002016365-A1 PYRAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS FOR MODULATING OR INHIBITING ERAB OR HADH2 ACTIVITY AGOURON PHARMACEUTICALS, INC. (US) 2002-02-28 WO claimed
US-20010036949-A1 Pharmaceutical composition and method of treatment of diseases of cognitive dysfunction in a mammal PFIZER PRODUCTS INC. 2001-11-01 US claimed
EP-1088550-A1 alpha-sulfonylamino hydroxamic acid inhibitors of matrix metallo-proteinases for the treatment of peripheral or central nervous system disorders Pfizer Products Inc. (US) 2001-04-04 EP claimed
WO-1998030243-A1 ACETYLCHOLINESTERASE INHIBITORS IN COMBINATION WITH MUSCARINIC AGONISTS FOR THE TREATMENT OF ALZHEIMER'S DISEASE WARNER-LAMBERT COMPANY (US) 1998-07-16 WO claimed