Rivastigmine

Rivastigmine

SCHEMBL29779663

CCN(C)C(=O)Oc1cccc([C@H](C)N(C)C)c1.O=C(O)[C@H](O)[C@@H](O)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBCHE

The experimentally established mechanism targets of Rivastigmine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 16/20 1.00
BCHE known ✓ P06276 11/20 1.00
MARK4 Q96L34 1/20 1.00
FAAH O00519 1/20 0.86
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rivastigmine SCHEMBL25232361 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL2763 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL3978590 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL29612619 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL30064255 1.00 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL13841811 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL29614698 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL1170429 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL6382107 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA
Rivastigmine SCHEMBL6382629 0.93 ACHE (1.00) ACHEBCHEMARK4FAAHMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260048083-A1 METHOD OF TREATING ALZHEIMER'S DISEASE WITH EXPANDED NATURAL KILLER CELLS NKMAX CO LTD (KR) 2026-02-19 US disclosed
EP-4674482-A2 PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF Otsuka Pharmaceutical Co., Ltd. (JP) 2026-01-07 EP disclosed
EP-4548926-A1 Y-SECRETASE INHIBITOR, AB-PEPTIDE PRODUCTION INHIBITOR, AND PHARMACEUTICAL Tohoku University (JP) 2025-05-07 EP disclosed
US-20250099459-A1 PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2025-03-27 US disclosed
WO-2024238387-A1 METHOD OF TREATING ALZHEIMER'S DISEASE WITH EXPANDED NATURAL KILLER CELLS NKMAX CO., LTD. (KR) 2024-11-21 WO disclosed
CN-118401123-A Brain function improving agent 国立大学法人大阪大学 2024-07-26 CN disclosed
WO-2024036005-A1 METHOD OF TREATING ALZHEIMER'S DISEASE WITH EXPANDED NATURAL KILLER CELLS NKMAX CO., LTD. (KR) 2024-02-15 WO disclosed
US-20230172880-A1 FAST-ACTING TOPICAL ANESTHETIC FORMULATIONS ACHELON, LLC 2023-06-08 US disclosed
EP-4138806-A1 FAST-ACTING TOPICAL ANESTHETIC FORMULATIONS Achelon, Inc. (US) 2023-03-01 EP disclosed
EP-3610879-B9 COMPOSITION FOR TREATMENT AND/OR PREVENTION OF ALZHEIMER'S DISEASE GLOVIA COMPANY LTD (JP) 2023-01-25 EP disclosed
US-20220370442-A1 PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2022-11-24 US disclosed
EP-3610879-B1 COMPOSITION FOR TREATMENT AND/OR PREVENTION OF ALZHEIMER'S DISEASE GLOVIA COMPANY LTD (JP) 2022-11-09 EP disclosed
CN-114712360-A Prophylactic and/or therapeutic agent comprising epiprazole or salt thereof 大塚制药株式会社 2022-07-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220370442-A1 PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF SLC6A3, SLC6A2, SNCA ACHE 104/4885BCHE 140/4885MARK4 409/4885
US-20250099459-A1 PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF SLC6A3, SLC6A2, SNCA ACHE 104/4885BCHE 140/4885MARK4 409/4885
US-20260048083-A1 METHOD OF TREATING ALZHEIMER'S DISEASE WITH EXPANDED NATURAL KILLER CELLS IL2, PBK, IL2RA ACHE 99/4885BCHE 126/4885MARK4 1550/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.