SCHEMBL27634604

SCHEMBL27634604

CC(CN)(C(N)=O)C(=O)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
MAPK1 P28482 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
KMT2A Q03164 2/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A3 Q01959 1/20 0.45
MMP8 P22894 1/20 0.44
TSHR P16473 2/20 0.42
CYP3A4 P08684 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 2/20 0.41
HCAR2 Q8TDS4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27615708 0.89 ALDH1A1 (0.51) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL27647172 0.86 KMT2A (0.50) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL23433097 0.85 ALDH1A1 (0.47) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL4178872 0.82 ALDH1A1 (0.55) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL21673204 0.81 ALDH1A1 (0.53) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL21673464 0.79 ALDH1A1 (0.51) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL29327822 0.79 ALDH1A1 (0.51) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL27615707 0.79 MMP8 (0.46) ALDH1A1KMT2AMMP8TSHRCYP3A4
SCHEMBL1809268 0.78 ALDH1A1 (0.58) ALDH1A1MAPK1L3MBTL1TDP1KMT2A
SCHEMBL19105239 0.78 ALDH1A1 (0.58) ALDH1A1MAPK1L3MBTL1TDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100413878-C Pyrazole derivatives, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof KISSEI PHARMACEUTICAL COMPANY (JP) 2008-08-27 CN disclosed
CN-100351263-C Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof KISSEI PHARMACEUTICAL COMPANY (JP) 2007-11-28 CN disclosed
CN-1688597-A Pyrazole derivatives, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof KISSEI PHARMACEUTICAL COMPANY (JP) 2005-10-26 CN disclosed
CN-1688596-A Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof KISSEI PHARMACEUTICAL COMPANY (JP) 2005-10-26 CN disclosed