SCHEMBL27635233

SCHEMBL27635233

C[C@@H]1C(O)=CC(=O)N1C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.43
KLK7 P49862 7/20 0.40
KDM4E B2RXH2 2/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
KLK5 Q9Y337 6/20 0.36
PRSS1 P07477 3/20 0.36
PRSS2 P07478 3/20 0.36
PRSS3 P35030 3/20 0.36
ELANE P08246 1/20 0.35
ALDH1A1 P00352 1/20 0.34
BCHE P06276 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
PIM1 P11309 1/20 0.32
PIM2 Q9P1W9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18593027 1.00 MAPK1 (0.43) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL31750269 0.82 KLK7 (0.36) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL34473806 0.82 KLK7 (0.36) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL16224738 0.80 KLK7 (0.40) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL22096754 0.77 KLK7 (0.40) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL34473950 0.76 KLK7 (0.35) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL10387166 0.76 KLK7 (0.40) MAPK1KLK7MAPTKLK5PRSS1
SCHEMBL28451513 0.75 KLK7 (0.40) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL21104039 0.75 KLK7 (0.40) MAPK1KLK7KDM4EMAPTTHRB
SCHEMBL13409204 0.74 USP2 (0.40) MAPK1KLK7KDM4EMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1688527-A Fused benzene derivatives and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2005-10-26 CN disclosed