SCHEMBL27637871

SCHEMBL27637871

Oc1ccc(C(F)(F)F)cc1-c1ccc2c(c1)OCO2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 1/20 0.52
GAPDH P04406 1/20 0.44
ALOX5 P09917 1/20 0.44
PTGS2 P35354 2/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
PTGS1 P23219 1/20 0.43
CLK1 P49759 1/20 0.42
CLK2 P49760 1/20 0.42
DYRK1A Q13627 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
CYP3A4 P08684 1/20 0.42
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 3/20 0.42
FABP4 P15090 1/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572292 0.77 ALOX5 (0.47) GAPDHALOX5PTGS2PTGS1CYP3A4
SCHEMBL14919902 0.77 AR (0.51) MAP2K4GAPDHALOX5CLK1CLK2
Hydrochloric Acid SCHEMBL6782247 0.76 ALOX5 (0.46) GAPDHALOX5PTGS2PTGS1CYP3A4
SCHEMBL1753671 0.75 PTGDR2 (0.65)
SCHEMBL27466656 0.74 BCL2L1 (0.59) GAPDHALOX5PTGS2PTGS1CYP3A4
SCHEMBL13247899 0.74 MAP2K4 (0.52) MAP2K4PTGS2PTGS1CLK1CLK2
SCHEMBL27541697 0.74 KIF11 (0.61) MAP2K4ALOX5KMT2AALDH1A1MEN1
SCHEMBL5098907 0.73 BCL2L1 (0.52) GAPDHALOX5KMT2AALDH1A1MEN1
SCHEMBL17141676 0.73 NTRK1 (0.45) KMT2AALDH1A1MEN1CYP1A2CYP2C19
SCHEMBL15675199 0.72 BIRC5 (0.44) AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100575330-C Novel compounds ASTRAZENECA AB 2009-12-30 CN claimed
CN-1791572-A Novel compounds ASTRAZENECA AB (SE) 2006-06-21 CN claimed
CN-100575330-C Novel compounds ASTRAZENECA AB 2009-12-30 CN disclosed
CN-1791572-A Novel compounds ASTRAZENECA AB (SE) 2006-06-21 CN disclosed