SCHEMBL27638465

SCHEMBL27638465

COc1cncn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.43
CYP11B2 P19099 4/20 0.43
CYP19A1 P11511 4/20 0.36
MAPK1 P28482 3/20 0.36
NR1I2 O75469 2/20 0.36
ADORA3 P0DMS8 2/20 0.36
TBXA2R P21731 2/20 0.36
CCKBR P32239 2/20 0.36
OPRK1 P41145 2/20 0.36
SLC6A3 Q01959 2/20 0.36
KCNH2 Q12809 2/20 0.36
NR1H4 Q96RI1 2/20 0.36
KCNN4 O15554 2/20 0.36
CYP3A4 P08684 2/20 0.36
RAB9A P51151 2/20 0.36
MEN1 O00255 1/20 0.36
SLC22A1 O15245 1/20 0.36
GMNN O75496 1/20 0.36
USP2 O75604 1/20 0.36
TRPM2 O94759 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27456864 0.79 CYP11B1 (0.40) CYP11B1CYP11B2CYP19A1MAPK1NR1I2
SCHEMBL16828671 0.79 CYP11B1 (0.40) CYP11B1CYP11B2CYP19A1KCNH2RAB9A
SCHEMBL16371592 0.77 CYP11B1 (0.47) CYP11B1CYP11B2CYP19A1MAPK1NR1I2
SCHEMBL4806085 0.77 CYP11B1 (0.43) CYP11B1CYP11B2CYP19A1MAPK1NR1I2
SCHEMBL21721462 0.74 TDP1 (0.32) TDP1
SCHEMBL6071929 0.73 CYP11B1 (0.35) CYP11B1CYP11B2
SCHEMBL6071924 0.73 CYP11B1 (0.35) CYP11B1CYP11B2
SCHEMBL2204500 0.73 CYP11B1 (0.43) CYP11B1CYP11B2CYP19A1MAPK1NR1I2
SCHEMBL11891091 0.71 CYP11B1 (0.39) CYP11B1CYP11B2CYP19A1MAPK1NR1I2
SCHEMBL20225762 0.70 FYN (0.32) CYP11B1CYP11B2FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101711242-B ((bicyclic heteroaryl) imidazolyl) methyl heteroaryl compounds as adrenergic receptor agonists ALLERGAN INC 2013-09-25 CN disclosed
CN-101743240-B ((phenyl) imidazolyl) methyl heteroaryl compounds ALLERGAN INC 2013-07-17 CN disclosed
CN-101743240-A ((phenyl) imidazolyl) methyl heteroaryl compounds ALLERGAN INC 2010-06-16 CN disclosed
CN-101711242-A ((bicyclic heteroaryl) imidazolyl) methyl heteroaryl compounds as adrenergic receptor agonists ALLERGAN INC 2010-05-19 CN disclosed
CN-1856475-A Isoquinoline potassium channel inhibitors MERCK & CO INC (US) 2006-11-01 CN disclosed