SCHEMBL27642201

SCHEMBL27642201

O=[N+]([O-])c1csc(-c2ccc(NC3=NCCN3)cc2)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 5/20 0.62
ADRA2A P08913 12/20 0.50
ADRA2B P18089 12/20 0.50
ADRA2C P18825 12/20 0.50
HTR1D P28221 1/20 0.50
HTR1B P28222 1/20 0.50
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977059 0.81 PTGIR (0.84) PTGIRADRA2AADRA2BADRA2CHTR1D
SCHEMBL27662722 0.79 PTGIR (0.58) PTGIRADRA2AADRA2BADRA2CADRA1D
SCHEMBL27662821 0.79 PTGIR (0.60) PTGIRADRA2AADRA2BADRA2CADRA1D
SCHEMBL5807468 0.77 PTGIR (1.00) PTGIRADRA2AADRA2BADRA2CHTR1D
SCHEMBL5827927 0.76 PTGIR (0.61) PTGIRADRA2AADRA2BADRA2CHTR1D
SCHEMBL28942366 0.74 PTGIR (0.64) PTGIRADRA2AADRA2BADRA2C
Acetic Acid SCHEMBL6967870 0.74 PTGIR (0.73) PTGIRADRA2AADRA2BADRA2CHTR1D
SCHEMBL27662630 0.72 ADRA2A (0.61) PTGIRADRA2AADRA2BADRA2C
SCHEMBL27642225 0.72 ADRA2A (0.52) PTGIRADRA2AADRA2BADRA2C
SCHEMBL27642292 0.70 ADRA2A (0.47) PTGIRADRA2AADRA2BADRA2CADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1849308-A Thiophenylaminoimidazolines ROCHE PALO ALTO LLC (CH) 2006-10-18 CN claimed
CN-1849308-A Thiophenylaminoimidazolines ROCHE PALO ALTO LLC (CH) 2006-10-18 CN disclosed