SCHEMBL27644451

SCHEMBL27644451

COc1ccc(C(C)C(C)CC(N)C(=O)O)c(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 3/20 0.43
GRIK2 Q13002 3/20 0.43
ADRA2A P08913 2/20 0.43
ADRA1A P35348 2/20 0.43
CYP2D6 P10635 1/20 0.43
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
TP53 P04637 1/20 0.41
KIF11 P52732 2/20 0.41
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
HSD17B10 Q99714 1/20 0.40
HTR2A P28223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27644642 0.90 ADRA1A (0.52) GRIK1GRIK2ADRA2AADRA1ACYP2D6
SCHEMBL27644165 0.88 TP53 (0.43) ADRA2AADRA1ACYP2D6MEN1MAPK1
SCHEMBL28758254 0.86 BCHE (0.41) GRIK1GRIK2ADRA2AADRA1ACYP2D6
SCHEMBL4989932 0.85 ADRA1A (0.45) ADRA2AADRA1ACYP2D6TP53HSD17B10
SCHEMBL27644169 0.83 MEN1 (0.39) GRIK1GRIK2CYP2D6MEN1KMT2A
SCHEMBL27665757 0.83 AKR1C3 (0.45) MEN1MAPK1KMT2ATP53HSD17B10
SCHEMBL27644290 0.82 GRIK1 (0.41) GRIK1GRIK2KIF11
SCHEMBL27665456 0.82 BCHE (0.44) GRIK1GRIK2ADRA2AADRA1ACYP2D6
SCHEMBL27665583 0.80 AOC3 (0.44) GRIK1GRIK2KIF11HSD17B10
SCHEMBL28815671 0.79 PTGS2 (0.46) ADRA2AADRA1ACYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1886363-A Amino acids with affinity for the alpha2delta-protein WARNER LAMBERT CO (US) 2006-12-27 CN claimed
CN-1886363-A Amino acids with affinity for the alpha2delta-protein WARNER LAMBERT CO (US) 2006-12-27 CN disclosed