SCHEMBL27645182

SCHEMBL27645182

FC(F)(F)Oc1ccc(CCCCCCC2CCN(c3ccnc4ccccc34)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NMT1 P30419 1/20 0.44
F10 P00742 2/20 0.43
GRM2 Q14416 2/20 0.42
KCNH2 Q12809 2/20 0.42
ADRB2 P07550 1/20 0.41
NCF1 P14598 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HRH3 Q9Y5N1 2/20 0.39
CHRM4 P08173 3/20 0.38
PDGFRB P09619 1/20 0.38
ACHE P22303 1/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27666211 1.00 NMT1 (0.44) NMT1F10GRM2KCNH2ADRB2
SCHEMBL28761502 0.87 KCNH2 (0.52) NMT1F10KCNH2ADRB2NCF1
SCHEMBL27644982 0.84 GRM2 (0.42) NMT1GRM2CHRM4ACHEDRD2
SCHEMBL2091985 0.83 GRM2 (0.45) NMT1GRM2CHRM4DRD2DRD4
SCHEMBL27645178 0.82 ADRB2 (0.51) NMT1F10KCNH2ADRB2NCF1
SCHEMBL2088412 0.82 GRM2 (0.41) NMT1GRM2CHRM4ACHEDRD2
SCHEMBL2093955 0.82 GRM2 (0.41) NMT1GRM2CHRM4ACHEDRD2
SCHEMBL28761490 0.80 NMT1 (0.49) NMT1KCNH2ADRB2NCF1MAPT
SCHEMBL2097669 0.80 GRM2 (0.44) GRM2CHRM4DRD2DRD4DRD3
SCHEMBL2093386 0.76 GRM2 (0.42) GRM2KCNH2CHRM4DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100497345-C 2, 3-dihydro-6-nitroimidazolo [2,1-b] oxazole compounds for the treatment of tuberculosis OTSUKA PHARMA CO LTD (JP) 2009-06-10 CN disclosed
CN-1878777-A 2,3-dihydro-6-nitroimidazo (2,1-b) oxazole compounds for the treatment of tuberculosis OTSUKA PHARMA CO LTD (JP) 2006-12-13 CN disclosed