SCHEMBL27645971

SCHEMBL27645971

CC(=O)Oc1ccc2cc(-c3n[nH]c4ccsc34)[nH]c2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 18/20 0.62
LCK P06239 3/20 0.62
TXK P42681 3/20 0.62
SYK P43405 3/20 0.62
CA2 P00918 1/20 0.46
PLK4 O00444 1/20 0.44
CHEK1 O14757 1/20 0.44
AURKA O14965 1/20 0.44
CCNB2 O95067 1/20 0.44
ABL1 P00519 1/20 0.44
CDK1 P06493 1/20 0.44
PDGFRB P09619 1/20 0.44
CDK4 P11802 1/20 0.44
SRC P12931 1/20 0.44
CCNB1 P14635 1/20 0.44
CCNA2 P20248 1/20 0.44
CCND1 P24385 1/20 0.44
CDK2 P24941 1/20 0.44
WEE1 P30291 1/20 0.44
TTK P33981 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2898497 0.90 ITK (0.59) ITKLCKTXKSYKPLK4
SCHEMBL1623341 0.80 ITK (0.63) ITKLCKTXKSYK
SCHEMBL2898022 0.79 ITK (0.47) ITKLCKTXKSYKPLK4
SCHEMBL27667060 0.79 ITK (0.61) ITKLCKTXKSYKPLK4
SCHEMBL1622165 0.78 ITK (0.54) ITKLCKTXKSYKPLK4
SCHEMBL16675978 0.77 ITK (1.00) ITKLCKTXKSYKPLK4
SCHEMBL2902831 0.77 ITK (0.45) ITKLCKTXKSYKAURKA
SCHEMBL2898574 0.77 ITK (0.45) ITKLCKTXKSYKPLK4
SCHEMBL12748758 0.76 ITK (0.64) ITKLCKTXKSYK
SCHEMBL27667096 0.76 ITK (0.64) ITKLCKTXKSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100398545-C Thienopyrazoles AVENTIS PHARMA INC (US) 2008-07-02 CN claimed
CN-1849322-A Thienopyrazoles AVENTIS PHARMA INC (US) 2006-10-18 CN claimed
CN-100398545-C Thienopyrazoles AVENTIS PHARMA INC (US) 2008-07-02 CN disclosed
CN-1849322-A Thienopyrazoles AVENTIS PHARMA INC (US) 2006-10-18 CN disclosed