SCHEMBL2902831

SCHEMBL2902831

O=C(NCCC1=CCCCC1)Oc1ccc2cc(-c3n[nH]c4ccsc34)[nH]c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.45
LCK P06239 2/20 0.45
TXK P42681 2/20 0.45
SYK P43405 2/20 0.45
AURKA O14965 1/20 0.41
HPGD P15428 3/20 0.40
ALDH1A1 P00352 7/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
TDP1 Q9NUW8 1/20 0.39
TP53 P04637 1/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
PRMT3 O60678 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.37
MCHR1 Q99705 1/20 0.37
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1623119 0.86 ITK (0.47) ITKLCKTXKSYKHPGD
SCHEMBL2898022 0.83 ITK (0.47) ITKLCKTXKSYKAURKA
SCHEMBL2898574 0.81 ITK (0.45) ITKLCKTXKSYKAURKA
SCHEMBL2903568 0.77 ITK (0.43) ITKLCKTXKSYKHPGD
SCHEMBL27645971 0.77 ITK (0.62) ITKLCKTXKSYKAURKA
SCHEMBL2903516 0.76 ITK (0.47) ITKLCKTXKSYKAURKA
SCHEMBL2898497 0.76 ITK (0.59) ITKLCKTXKSYKAURKA
SCHEMBL13869803 0.69 ITK (0.60) ITKLCKTXKSYKALDH1A1
SCHEMBL1622884 0.69 ITK (0.50) ITKLCKTXKSYKHPGD
SCHEMBL27667096 0.68 ITK (0.64) ITKLCKTXKSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682553-B1 THIENOPYRAZOLES AVENTIS PHARMA INC (US) 2010-05-19 EP claimed