SCHEMBL27652199

SCHEMBL27652199

O=S(=O)(OCC(F)c1ccccc1)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.39
CA1 P00915 3/20 0.37
NPSR1 Q6W5P4 2/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35
CA7 P43166 1/20 0.35
HSD11B1 P28845 2/20 0.34
CYP2C19 P33261 1/20 0.33
SLC6A4 P31645 1/20 0.33
TACR1 P25103 2/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33
CACNA1C Q13936 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31362703 0.84 NPSR1 (0.44) CA2CA1NPSR1ALDH1A1MAPT
SCHEMBL5925000 0.81 TAAR1 (0.41) CA2CA1TACR1
SCHEMBL5925006 0.81 TAAR1 (0.41) CA2CA1TACR1
SCHEMBL4131267 0.80 SRC (0.40) CA2CA1NPSR1ALDH1A1MAPT
SCHEMBL11044378 0.80 CA1 (0.36) CA2CA1NPSR1MAPTKMT2A
Alcohol SCHEMBL11044375 0.75 LMNA (0.35) NPSR1ALDH1A1MAPTKMT2ACYP2C19
SCHEMBL16563079 0.74 CA2 (0.45) CA2CA1CA9CYP1A2
SCHEMBL12012235 0.72 CA2 (0.44) CA2CA1NPSR1ALDH1A1MAPK1
SCHEMBL19713389 0.72 CA2 (0.44) CA2CA1NPSR1ALDH1A1MAPK1
SCHEMBL12012234 0.72 CA2 (0.44) CA2CA1NPSR1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102329267-A 6-substituted 2,3,4, 5-tetrahydro-1H-benzo [d] aza as 5-HT2Creceptor agonists LILLY CO ELI 2012-01-25 CN disclosed
CN-102311387-A 6-substituted 2,3,4, 5-tetrahydro-1H-benzo [d] aza as 5-HT2Creceptor agonists LILLY CO ELI 2012-01-11 CN disclosed
CN-1934088-A As 5-HT2c6-substituted 2,3,4, 5-tetrahydro-1H-benzo [ d ] receptor agonists]Aza * LILLY CO ELI (US) 2007-03-21 CN disclosed