SCHEMBL27655822

SCHEMBL27655822

O=C(NNCl)c1ccncc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.75
TP53 P04637 1/20 0.62
CA1 P00915 1/20 0.58
CA9 Q16790 1/20 0.58
MAOA P21397 1/20 0.58
MAOB P27338 1/20 0.58
PTGS2 P35354 1/20 0.58
KDM4E B2RXH2 1/20 0.57
MPO P05164 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
ADORA3 P0DMS8 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2A6 P11509 1/20 0.57
CYP2C19 P33261 1/20 0.57
GAA P10253 1/20 0.55
HPGD P15428 2/20 0.53
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MAPK1 P28482 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2992964 0.86 ALDH1A1 (1.00) ALDH1A1TP53CA1CA9MAOA
SCHEMBL28791700 0.82 ALDH1A1 (0.67) ALDH1A1TP53CA1CA9MAOA
SCHEMBL2988323 0.80 ALDH1A1 (0.86) ALDH1A1TP53CA1CA9MAOA
SCHEMBL3003252 0.79 ALDH1A1 (0.69) ALDH1A1TP53CA1CA9MAOA
SCHEMBL25738324 0.78 ALDH1A1 (0.75) ALDH1A1TP53CA1CA9MAOA
SCHEMBL2995413 0.78 ALDH1A1 (0.75) ALDH1A1TP53CA1CA9MAOA
SCHEMBL27895863 0.78 ALDH1A1 (0.75) ALDH1A1TP53CA1CA9MAOA
SCHEMBL2986200 0.78 ALDH1A1 (0.83) ALDH1A1TP53CA1CA9MAOA
SCHEMBL3000231 0.78 ALDH1A1 (0.83) ALDH1A1TP53CA1CA9MAOA
SCHEMBL3935111 0.77 ALDH1A1 (0.79) ALDH1A1TP53CA1CA9MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101723941-A “1,2,4” oxadiazole as a metabotropic glutamate receptor-5 modulator ASTRAZENECA AB 2010-06-09 CN disclosed
CN-101096368-A Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists NPS PHARMA INC (SE) 2008-01-02 CN disclosed
CN-1984907-A Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists ASTRAZENECA AB (SE) 2007-06-20 CN disclosed
CN-1894241-A \"1, 2, 4\" oxadiazoles as modulators of metabotropic glutamate receptor-5 ASTRAZENECA AB (SE) 2007-01-10 CN disclosed