SCHEMBL276571

SCHEMBL276571

O=C(O)C(Cc1ccc(O)cc1)N(Br)Br

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.55
FOLH1 Q04609 1/20 0.45
NAALAD2 Q9Y3Q0 1/20 0.45
CA2 P00918 1/20 0.44
CAMK2A Q9UQM7 1/20 0.44
ESR1 P03372 4/20 0.43
ESR2 Q92731 4/20 0.43
POLB P06746 1/20 0.43
TAAR1 Q96RJ0 3/20 0.41
SLC6A2 P23975 1/20 0.41
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
TRPV1 Q8NER1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL276572 1.00 SLC7A5 (0.55) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL29278381 0.98 SLC7A5 (0.53) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL23610314 0.86 SLC7A5 (0.51) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL23610302 0.86 SLC7A5 (0.51) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL31092852 0.85 CYP1A2 (0.55) SLC7A5FOLH1NAALAD2
SCHEMBL2986794 0.83 SLC7A5 (0.56) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL2542276 0.83 SLC7A5 (0.56) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL6300612 0.83 SLC7A5 (0.53) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL6300611 0.83 SLC7A5 (0.53) SLC7A5FOLH1NAALAD2CA2CAMK2A
SCHEMBL38225 0.81 SLC7A5 (0.55) SLC7A5FOLH1CA2CAMK2AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 199 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116574138-B Dibromotyrosine-iridium complex and preparation method and application thereof 广东医科大学 2024-01-26 CN claimed
CN-116574138-A Dibromotyrosine-iridium complex and preparation method and application thereof 广东医科大学 2023-08-11 CN claimed
CN-109988312-B Polyamide acid ester, preparation method, negative polyimide composition and application 深圳先进技术研究院 2023-04-11 CN claimed
CN-107523219-B Chemical Mechanical Polishing (CMP) of cobalt-containing substrates 弗萨姆材料美国有限责任公司 2020-12-29 CN claimed
US-10745589-B2 Chemical mechanical polishing (CMP) of cobalt-containing substrate VERSUM MATERIALS US, LLC (US) 2020-08-18 US claimed
EP-3257910-B1 CHEMICAL MECHANICAL POLISHING (CMP) COMPOSITION, METHOD AND SYSTEM FOR COBALT-CONTAINING SUBSTRATE VERSUM MAT US LLC (US) 2019-03-27 EP claimed
US-20170362466-A1 Chemical Mechanical Polishing (CMP) of Cobalt-Containing substrate VERSUM MATERIALS US, LLC (US) 2017-12-21 US claimed
EP-3257910-A1 CHEMICAL MECHANICAL POLISHING (CMP) COMPOSITION, METHOD AND SYSTEM FOR COBALT-CONTAINING SUBSTRATE Versum Materials US, LLC (US) 2017-12-20 EP claimed
CN-105873944-A Pro-angiogenic peptides and peptide conjugates 耶路撒冷希伯来大学伊森姆研究发展有限公司 2016-08-17 CN claimed
EP-1856274-B1 SYSTEMIC MARKERS FOR ASTHMA AND ANALOGOUS DISEASES CLEVELAND CLINIC FOUNDATION (US) 2014-08-27 EP claimed
US-6841689-B2 Process using catalyst comprising soluble polymer and polymino acid STYLACATS LIMITED (GB) 2005-01-11 US claimed
US-20040048739-A1 Catalyst comprising soluble polymer and polymino acid STYLACATS LIMITED (GB) 2004-03-11 US claimed
US-20030207324-A1 IMMUNOTHERAPY BY MODULATION OF ANTIGEN PRESENTATION HUMPHREYS ROBERT E 2003-11-06 US claimed
EP-1289974-A1 CATALYST COMPRISING SOLUBLE POLYMER AND POLYAMINO ACID Stylacats Ltd (GB) 2003-03-12 EP claimed
US-20020048775-A1 Diagnostic methods for asthma NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2002-04-25 US claimed
WO-2001094327-A1 CATALYST COMPRISING SOLUBLE POLYMER AND POLYAMINO ACID STYLACATS LIMITED (GB) 2001-12-13 WO claimed
US-6306576-B1 ANALYZING SAMPLE FOR 3-BROMOTYROSINE AND/OR 3,5-DIBROMOTYROSINE; ELEVATED LEVELS INDICATE DISEASE ASSOCIATED WITH ACTIVATED EOSINOPHILS CLEVELAND CLINIC FOUNDATION 2001-10-23 US claimed
US-5919639-A INCUBATING MAJOR HISTOCOMPATIBILITY COMPLEX CLASS II EXPRESSING ANTIGEN PRESENTING CELL WITH MAMMALIAN INVARIANT CHAIN PEPTIDE OF 4-16 AMINO ACIDS, A MAJOR HISTOCOMPATIBILITY COMPLEX CLASS II RESTRICTED ANTIGENIC PEPTIDE, AND A T CELL UNIVERSITY OF MASSACHUSETTS (US) 1999-07-06 US claimed
US-5756650-A COMPOSITION COMPRISING POLYAMIC ACID, CURE ACCELERATOR SELECTED FROM GROUP CONSISTING OF NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AMINO ACID COMPOUND, AROMATIC COMPOUND HAVING TWO OR MORE HYDROXYL GROUPS KABUSHIKI KAISHA TOSHIBA (JP) 1998-05-26 US claimed
WO-1997049430-A1 IMMUNOTHERAPY BY MODULATION OF ANTIGEN PRESENTATION ANTIGEN EXPRESS, INC. (US) 1997-12-31 WO claimed