SCHEMBL27657161

SCHEMBL27657161

CN1CCC(c2ccc(-c3ccnc(NC4CC(C)(C)NC(C)(C)C4)n3)s2)CC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 4/20 0.47
CDK4 P11802 4/20 0.45
CCND1 P24385 4/20 0.45
CDK2 P24941 3/20 0.45
CDK1 P06493 2/20 0.45
CCNB1 P14635 2/20 0.45
CCNA2 P20248 2/20 0.45
CCNA1 P78396 2/20 0.45
RET P07949 1/20 0.45
CCND3 P30281 2/20 0.44
CDK6 Q00534 2/20 0.44
MAPK8 P45983 2/20 0.42
KCNH2 Q12809 2/20 0.42
MAPK10 P53779 2/20 0.41
MAPK9 P45984 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
CCNE1 P24864 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3476963 0.83 KCNH2 (0.35) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL3478504 0.83 IKBKB (0.41) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL4491192 0.80 IKBKB (0.41) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL4487841 0.80 KCNH2 (0.40) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL16199971 0.80 KCNH2 (0.41) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL4484036 0.79 KCNH2 (0.35) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL4491170 0.79 KCNH2 (0.35) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL3470774 0.78 CDK9 (0.40) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL3478098 0.78 LMNA (0.41) IKBKBCDK4CCND1CDK2CDK1
SCHEMBL3477653 0.78 KCNH2 (0.43) CDK4CCND1CDK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1802357-A 2-aminopyrimidine derivatives and their medical use NOVARTIS AG (CH) 2006-07-12 CN disclosed