SCHEMBL27664302

SCHEMBL27664302

CSC[C@@H]1CCCN1.O=COCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
LTA4H P09960 5/20 0.42
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
KHK P50053 1/20 0.39
GHSR Q92847 2/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
TSHR P16473 1/20 0.38
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27825232 0.85 TSHR (0.49) POLBLTA4HHTR2CHTR2BGHSR
SCHEMBL28776632 0.82 POLB (0.52) POLBLTA4HGHSRTSHR
SCHEMBL28270587 0.81 TSHR (0.46) POLBHTR2CHTR2BTSHR
SCHEMBL27843143 0.77 HTR2C (0.42) POLBLTA4HHTR2CHTR2BGHSR
SCHEMBL28238992 0.75 TSHR (0.48) POLBHTR2CTSHR
SCHEMBL27772138 0.74 TSHR (0.43) POLBHTR2CTSHR
Azetidine SCHEMBL27976635 0.74 TSHR (0.41) HTR2CTSHR
SCHEMBL27879042 0.74 CTSC (0.41) POLBLTA4HHTR2CHTR2BTSHR
SCHEMBL27873296 0.72 TSHR (0.46) TSHR
SCHEMBL23251393 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1852712-B Dual NK1/NK3 antagonists for treating schizophrenia HOFFMANN LA ROCHE 2010-06-09 CN disclosed
CN-1852712-A Dual NK1/NK3 antagonists for treating schizophrenia HOFFMANN LA ROCHE (CH) 2006-10-25 CN disclosed