SCHEMBL27825232

SCHEMBL27825232

CC1CCCN1.O=COCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
POLB P06746 1/20 0.44
HTR2C P28335 2/20 0.43
HTR2B P41595 1/20 0.43
LTA4H P09960 2/20 0.40
GLA P06280 1/20 0.37
CTSC P53634 1/20 0.37
GHSR Q92847 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28270587 0.92 TSHR (0.46) TSHRPOLBHTR2CHTR2BGLA
SCHEMBL27664302 0.85 POLB (0.43) TSHRPOLBHTR2CHTR2BLTA4H
SCHEMBL27843143 0.85 HTR2C (0.42) TSHRPOLBHTR2CHTR2BLTA4H
SCHEMBL28238992 0.82 TSHR (0.48) TSHRPOLBHTR2CGLA
Azetidine SCHEMBL27976635 0.82 TSHR (0.41) TSHRHTR2C
SCHEMBL27772138 0.82 TSHR (0.43) TSHRPOLBHTR2C
SCHEMBL28776632 0.82 POLB (0.52) TSHRPOLBLTA4HGHSR
SCHEMBL27879042 0.82 CTSC (0.41) TSHRPOLBHTR2CHTR2BLTA4H
SCHEMBL27939939 0.81 TSHR (0.42) TSHRHTR2CLTA4HGLA
SCHEMBL28274307 0.81 TSHR (0.42) TSHRHTR2CLTA4HGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101998959-B Benzoxazole carboxamide inhibitors of poly(ADP-ribose)polymerase (PARP) BIOMARIN PHARM INC 2013-08-28 CN disclosed
CN-101998959-A Benzoxazole carboxamide inhibitors of poly(ADP-ribose)polymerase (PARP) LEAD THERAPEUTICS INC 2011-03-30 CN disclosed