SCHEMBL27664997

SCHEMBL27664997

NCc1ccccc1-c1cc(N2CCOCC2)nc(Cl)c1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 7/20 0.44
HTT P42858 4/20 0.43
LMNA P02545 3/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
PIK3CA P42336 5/20 0.43
MAPT P10636 1/20 0.42
NAPEPLD Q6IQ20 1/20 0.41
PIK3CD O00329 4/20 0.41
PIK3CG P48736 4/20 0.41
PKM P14618 1/20 0.41
PIK3C2B O00750 1/20 0.41
MTOR P42345 1/20 0.41
AKT1 P31749 1/20 0.40
RAB9A P51151 1/20 0.39
ATM Q13315 1/20 0.39
CNR2 P34972 1/20 0.39
POLB P06746 2/20 0.39
GBA1 P04062 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399406 0.86 MAPT (0.49) PIK3CBHTTLMNAKDM4EALDH1A1
SCHEMBL27684509 0.78 CNR2 (0.43) PIK3CBHTTLMNAKDM4EALDH1A1
SCHEMBL27664989 0.70 DPP4 (0.47) POLBHSD17B10
SCHEMBL7216508 0.68 CNR2 (0.58) HTTLMNARAB9ACNR2POLB
SCHEMBL17476483 0.68 ALDH1A1 (0.43) PIK3CBHTTLMNAKDM4EALDH1A1
SCHEMBL27882082 0.67 CYP2C19 (0.45) PIK3CBHTTLMNAKDM4EALDH1A1
SCHEMBL3095284 0.67 IKBKB (0.56) PIK3CBHTTKDM4EALDH1A1HPGD
SCHEMBL2130081 0.67 KMT2A (0.54) HTTKDM4EALDH1A1HPGDPIK3CA
SCHEMBL1239649 0.67 KDM4E (0.66) PIK3CBHTTLMNAKDM4EALDH1A1
SCHEMBL27967258 0.65 KMT2A (0.49) PIK3CBHTTLMNAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1984891-B Process for the preparation of carboxamide pyridine derivatives useful as intermediates in the synthesis of NK-1 receptor antagonists HOFFMANN LA ROCHE 2012-08-08 CN disclosed
CN-1984891-A Process for the preparation of carboxamide pyridine derivatives useful as intermediates in the synthesis of NK-1 receptor antagonists HOFFMANN LA ROCHE (CH) 2007-06-20 CN disclosed