SCHEMBL27666271

SCHEMBL27666271

Clc1cccc(CN2CCN(c3cccc4ncccc34)CC2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.55
NCF1 P14598 1/20 0.52
HTR6 P50406 1/20 0.49
DRD3 P35462 2/20 0.49
CYP3A4 P08684 1/20 0.49
CHRM1 P11229 1/20 0.49
OPRK1 P41145 1/20 0.49
PDE4D Q08499 1/20 0.49
KCNH2 Q12809 1/20 0.49
PDE3A Q14432 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
RAD52 P43351 1/20 0.47
GPR6 P46095 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
FAAH O00519 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401253 0.81 KCNH2 (0.64) SIGMAR1NCF1KCNH2MAPTDRD4
SCHEMBL27470939 0.78 CYP3A4 (0.57) NCF1DRD3CYP3A4CHRM1OPRK1
SCHEMBL27470403 0.78 CYP3A4 (0.71) NCF1DRD3CYP3A4CHRM1OPRK1
SCHEMBL27666154 0.77 KCNH2 (0.54) NCF1DRD3CYP3A4CHRM1OPRK1
SCHEMBL13987031 0.77 NR4A1 (0.55) NCF1DRD3KCNH2MAPTDRD2
SCHEMBL13987033 0.74 KCNH2 (0.61) HTR6DRD3CYP3A4KCNH2HRH3
SCHEMBL8130723 0.74 SIGMAR1 (0.58) SIGMAR1HTR6MAPTTSHRDRD4
SCHEMBL2165351 0.74 DHFR (0.62) SIGMAR1NCF1DRD3MAPTTSHR
SCHEMBL8173934 0.74 SIGMAR1 (0.70) SIGMAR1DRD3MAPTTSHRDRD2
SCHEMBL9229789 0.73 KCNH2 (0.60) DRD3CYP3A4CHRM1OPRK1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100497345-C 2, 3-dihydro-6-nitroimidazolo [2,1-b] oxazole compounds for the treatment of tuberculosis OTSUKA PHARMA CO LTD (JP) 2009-06-10 CN disclosed
CN-1878777-A 2,3-dihydro-6-nitroimidazo (2,1-b) oxazole compounds for the treatment of tuberculosis OTSUKA PHARMA CO LTD (JP) 2006-12-13 CN disclosed