SCHEMBL27667163

SCHEMBL27667163

CC(C)(Cc1c(C(N)=O)c(=O)[nH]c2cc(Cc3ccc(F)cc3C(F)(F)F)cnc12)C(O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 4/20 0.34
CYP3A4 P08684 4/20 0.34
PGR P06401 2/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
P2RX7 Q99572 2/20 0.33
SLC6A4 P31645 5/20 0.33
SLC6A2 P23975 4/20 0.33
PARP1 P09874 3/20 0.32
PARP2 Q9UGN5 3/20 0.32
PARP6 Q2NL67 2/20 0.32
PARP3 Q9Y6F1 2/20 0.32
TNKS O95271 1/20 0.32
BTK Q06187 1/20 0.31
SLC6A3 Q01959 1/20 0.31
DHFR P00374 1/20 0.31
MAPK1 P28482 1/20 0.31
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27686147 0.90 HDAC3 (0.34) HDAC3HDAC1HDAC2HDAC6P2RX7
SCHEMBL27667166 0.82 NTRK1 (0.32) PARP1PARP2PARP6PARP3TNKS
SCHEMBL5547490 0.77 HDAC3 (0.37) HDAC3HDAC1HDAC2HDAC6P2RX7
SCHEMBL5546928 0.74 TDP1 (0.36) HDAC3HDAC1HDAC2HDAC6P2RX7
SCHEMBL27666982 0.74 BTK (0.34) PARP1PARP2PARP6PARP3TNKS
SCHEMBL27667160 0.74 GRM2 (0.34) PARP1PARP2PARP6PARP3TNKS
SCHEMBL27667159 0.74 HDAC3 (0.35) HDAC3HDAC1HDAC2HDAC6P2RX7
SCHEMBL5546798 0.73 GPR52 (0.38) HDAC3HDAC1HDAC2HDAC6P2RX7
SCHEMBL5540956 0.73 TDP1 (0.40) HDAC3HDAC1HDAC2HDAC6P2RX7
SCHEMBL27667170 0.73 BTK (0.33) PARP1PARP2PARP6PARP3TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed