SCHEMBL27667166

SCHEMBL27667166

NC(=O)c1c(CC(O)N2CCOCC2)c2ncc(Cc3ccc(F)cc3C(F)(F)F)cc2[nH]c1=O

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 3/20 0.32
PARP1 P09874 7/20 0.32
PARP2 Q9UGN5 3/20 0.32
PARP6 Q2NL67 2/20 0.32
PARP3 Q9Y6F1 2/20 0.32
TNKS O95271 1/20 0.32
PIK3CA P42336 1/20 0.30
GRIN2B Q13224 1/20 0.30
XIAP P98170 1/20 0.30
HTR2C P28335 1/20 0.30
MCHR1 Q99705 1/20 0.30
TRPC5 Q9UL62 1/20 0.30
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27666972 0.88 NTRK1 (0.36) NTRK1PARP1PARP2PARP6PARP3
SCHEMBL27686147 0.87 HDAC3 (0.34) PARP1PARP2PARP6PARP3TNKS
SCHEMBL27667163 0.82 NR3C1 (0.34) PARP1PARP2PARP6PARP3TNKS
SCHEMBL5545421 0.76 PARP1 (0.47) PARP1
SCHEMBL5545347 0.74 KDM4E (0.51) PARP1
SCHEMBL27667070 0.74 NTRK1 (0.36) NTRK1PARP1PARP2PARP6PARP3
SCHEMBL27666982 0.73 BTK (0.34) PARP1PARP2PARP6PARP3TNKS
SCHEMBL27667206 0.71 SCN9A (0.36)
SCHEMBL5547490 0.70 HDAC3 (0.37) PARP1NR1H2NR1H3
SCHEMBL27686339 0.70 NTRK1 (0.33) NTRK1PARP1PIK3CAGRIN2BXIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed