SCHEMBL27667635

SCHEMBL27667635

O=Cc1nccc2ccccc12.[H+]

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.48
CYP2A6 P11509 2/20 0.48
F12 P00748 1/20 0.48
NCF1 P14598 1/20 0.48
NOS3 P29474 1/20 0.48
NOS1 P29475 1/20 0.48
NOS2 P35228 1/20 0.48
BACE1 P56817 1/20 0.48
S100A4 P26447 1/20 0.47
NQO2 P16083 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.46
MAPT P10636 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP3A4 P08684 3/20 0.43
LMNA P02545 2/20 0.43
APEX1 P27695 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL194555 0.98 PLAU (0.50) PLAUCYP2A6F12NCF1NOS3
Hydrochloric Acid SCHEMBL27892483 0.96 PLAU (0.48) PLAUCYP2A6F12NCF1NOS3
Formaldehyde SCHEMBL22343884 0.94 PLAU (0.47) PLAUCYP2A6F12NCF1NOS3
Boric Acid SCHEMBL27989300 0.91 NCOA3 (0.47) PLAUCYP2A6F12NCF1NOS3
Furan SCHEMBL28122491 0.89 S100A4 (0.43) PLAUCYP2A6F12NCF1NOS3
Quinoline SCHEMBL28086932 0.86 ALDH1A1 (0.55) PLAUCYP2A6F12NCF1NOS3
Quinazoline SCHEMBL28491213 0.81 EGFR (0.57) PLAUCYP2A6F12NCF1NOS3
Quinoline SCHEMBL28123047 0.80 ALDH1A1 (0.47) PLAUCYP2A6F12NCF1NOS3
SCHEMBL25376432 0.79 S100A4 (0.39) PLAUCYP2A6F12NCF1NOS3
SCHEMBL895053 0.78 PLAU (0.50) PLAUCYP2A6F12NCF1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107382858-A The serial assimilation compound of 1,2,3,4 tetrahydroisoquinoline 4 and its synthetic method and application 天津师范大学 2017-11-24 CN claimed
CN-101602725-B Synthetic method of hexahydroisoquinoline-1-keto compound UNIV ZHEJIANG 2012-07-11 CN claimed
CN-101602725-A Hexahydroisoquinolin--1-keto compound and synthetic method thereof UNIV ZHEJIANG (CN) 2009-12-16 CN claimed
CN-110003274-A Phosphonylation dihydro-isoquinoline ketone compounds and preparation method thereof 郑州大学 2019-07-12 CN disclosed
CN-107778238-A A kind of new synthetic method of the ketone of 3,4 dihydro-isoquinoline 1 and isoindoline 1 ketone derivatives 中山大学 2018-03-09 CN disclosed
CN-102124000-B Pyridine compounds ASTRAZENECA AB 2014-09-17 CN disclosed
CN-101602725-B Synthetic method of hexahydroisoquinoline-1-keto compound UNIV ZHEJIANG 2012-07-11 CN disclosed
CN-102124000-A Pyridine compounds ASTRAZENECA AB 2011-07-13 CN disclosed
CN-101602725-A Hexahydroisoquinolin--1-keto compound and synthetic method thereof UNIV ZHEJIANG (CN) 2009-12-16 CN disclosed
CN-101602725-A Hexahydroisoquinolin--1-keto compound and synthetic method thereof UNIV ZHEJIANG (CN) 2009-12-16 CN disclosed
CN-101151250-A Processes for preparing morphinans and intermediates thereof MALLINCKRODT INC (US) 2008-03-26 CN disclosed
CN-1913778-A Aminocyclopentyl pyridopyrazinone modulators of chemokine receptor activity MERCK & CO INC (US) 2007-02-14 CN disclosed