SCHEMBL27670397

SCHEMBL27670397

CC(C)(C)OOC(=O)c1ccc(N2CC[C@H](N)C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
GPR119 Q8TDV5 5/20 0.44
NAMPT P43490 1/20 0.43
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
PIM1 P11309 1/20 0.40
CLK2 P49760 1/20 0.40
MAP4K2 Q12851 1/20 0.40
CAMK2D Q13557 1/20 0.40
DYRK1A Q13627 1/20 0.40
PIM3 Q86V86 1/20 0.40
AURKB Q96GD4 1/20 0.40
PRKD2 Q9BZL6 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
STK17A Q9UEE5 1/20 0.40
MAP4K5 Q9Y4K4 1/20 0.40
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27670398 1.00 ALDH1A1 (0.47) ALDH1A1TSHRHSD17B10TDP1GPR119
SCHEMBL2409983 0.87 GPR119 (0.51) ALDH1A1GPR119NAMPTPRKD3MAP4K4
SCHEMBL2409985 0.87 GPR119 (0.51) ALDH1A1GPR119NAMPTPRKD3MAP4K4
SCHEMBL27785053 0.82 ALDH1A1 (0.44) ALDH1A1TSHRHSD17B10TDP1GPR119
SCHEMBL4833816 0.82 ALDH1A1 (0.55) ALDH1A1TSHRHSD17B10NAMPTPRKD3
SCHEMBL14155927 0.82 ALDH1A1 (0.55) ALDH1A1TSHRHSD17B10NAMPTPRKD3
SCHEMBL28879095 0.80 ALDH1A1 (0.47) ALDH1A1TSHRHSD17B10TDP1GPR119
SCHEMBL382516 0.79 PRKD3 (0.56) ALDH1A1TSHRTDP1PRKD3MAP4K4
SCHEMBL383362 0.79 PRKD3 (0.56) ALDH1A1TSHRTDP1PRKD3MAP4K4
SCHEMBL5207933 0.79 GPR119 (0.56) ALDH1A1GPR119MAPTUSP2SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101679239-B Inhibitors of histone deacetylase METHYLGENE INC 2014-12-10 CN disclosed
CN-1997649-B Inhibitors of histone deacetylase METHYLGENE INC 2010-08-11 CN disclosed
CN-101679239-A inhibitors of histone deacetylase METHYLGENE INC 2010-03-24 CN disclosed
CN-1997649-A Inhibitors of histone deacetylase METHYLGENE INC (CA) 2007-07-11 CN disclosed