SCHEMBL27670535

SCHEMBL27670535

CC1=C(C(N)=O)SC(C)N1c1cccc(C(O)CN2CCN(c3cccc4nc(C)ccc34)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 17/20 0.43
HTR1D P28221 17/20 0.43
HTR1B P28222 17/20 0.43
DRD2 P14416 8/20 0.42
HTR7 P34969 8/20 0.42
DRD3 P35462 8/20 0.42
KCNH2 Q12809 7/20 0.42
HTR2A P28223 7/20 0.42
HTR2B P41595 7/20 0.42
HTR6 P50406 2/20 0.42
HTR2C P28335 6/20 0.42
CYP2C9 P11712 2/20 0.42
ADRA1A P35348 3/20 0.42
CYP3A4 P08684 2/20 0.42
SLC6A4 P31645 1/20 0.42
ADRB2 P07550 2/20 0.41
ADRB1 P08588 2/20 0.41
ADRB3 P13945 2/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1B P35368 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27650461 0.99 ADRA1A (0.42) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL27670574 0.92 HTR1A (0.44) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL27650450 0.85 HTR1A (0.61) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL2884411 0.79 HTR1A (0.65) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL2884192 0.77 HTR1D (0.54) HTR1AHTR1DHTR1BDRD2HTR7
SCHEMBL27650507 0.77 HTR1D (0.53) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL2885896 0.76 HTR1D (0.69) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL2884177 0.76 HTR1D (0.53) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL2884542 0.76 HTR1A (0.68) HTR1AHTR1DHTR1BDRD2HTR7
Hydrochloric Acid SCHEMBL27650488 0.76 HTR1A (0.56) HTR1AHTR1DHTR1BDRD2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100441571-C Quinoline and quinazoline derivatives having affinity for 5HT1-type receptors GLAXO GROUP LTD (GB) 2008-12-10 CN claimed
CN-1852896-A Quinoline and quinazoline derivatives having affinity for 5HT 1-type receptors GLAXO GROUP LTD (GB) 2006-10-25 CN claimed
CN-100441571-C Quinoline and quinazoline derivatives having affinity for 5HT1-type receptors GLAXO GROUP LTD (GB) 2008-12-10 CN disclosed
CN-1852896-A Quinoline and quinazoline derivatives having affinity for 5HT 1-type receptors GLAXO GROUP LTD (GB) 2006-10-25 CN disclosed