SCHEMBL27670844

SCHEMBL27670844

CCn1cnc2c(=O)n(-c3ccc(F)cc3)c(C(S)c3csc(C(F)(F)F)n3)nc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
LMNA P02545 2/20 0.34
HPGD P15428 2/20 0.34
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CDK1 P06493 5/20 0.33
ALDH1A1 P00352 1/20 0.33
DGKZ Q13574 3/20 0.33
UBE2M P61081 1/20 0.32
DCUN1D1 Q96GG9 1/20 0.32
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27670874 0.85 CDK1 (0.33) NPC1RAB9ALMNAHPGDTSHR
SCHEMBL27670851 0.81 POLB (0.33) PDE4APDE4BPDE4CPDE4DMCHR1
SCHEMBL27670909 0.79 CNR1 (0.35) NPC1TSHRPDE4APDE4BPDE4C
SCHEMBL5428540 0.78 MEN1 (0.38) NPC1RAB9ALMNAHPGDTSHR
SCHEMBL4525582 0.74 CDK1 (0.38) NPC1RAB9ALMNAHPGDTSHR
SCHEMBL4506865 0.73 CDK1 (0.40) CDK1CXCR3
SCHEMBL2233449 0.72 MAT2A (0.42) NPC1RAB9ALMNAHPGDTSHR
SCHEMBL5431647 0.72 NPSR1 (0.38) LMNATSHRSMN1; SMN2ALDH1A1
SCHEMBL4978987 0.71 SMN1; SMN2 (0.37) NPC1RAB9ALMNAHPGDTSHR
SCHEMBL5427488 0.70 CNR1 (0.33) NPC1TSHRSMN1; SMN2PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1902201-A Bicyclic pyrimidin-4-(3H)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (VR1) MERCK SHARP & DOHME (GB) 2007-01-24 CN claimed
CN-1902201-A Bicyclic pyrimidin-4-(3H)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (VR1) MERCK SHARP & DOHME (GB) 2007-01-24 CN disclosed