SCHEMBL27670909

SCHEMBL27670909

CCn1cnc2c(=O)n(-c3ccc(Cl)cc3)c(C(S)c3nc(C(F)(F)F)cs3)nc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.35
FFAR2 O15552 1/20 0.32
POLB P06746 1/20 0.31
HIF1A Q16665 1/20 0.31
MAT2A P31153 1/20 0.31
TSHR P16473 2/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
NPC1 O15118 1/20 0.31
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30
GRM1 Q13255 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27670874 0.93 CDK1 (0.33) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL27670910 0.89 FFAR2 (0.32) CNR1FFAR2POLBMAT2AGRM1
SCHEMBL27650758 0.79 AKR1B1 (0.36) CNR1POLBHIF1AMAT2ATSHR
SCHEMBL27670844 0.79 NPC1 (0.34) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL5446891 0.78 CNR1 (0.38) CNR1HIF1AMAT2ATSHRPDE4A
SCHEMBL4516843 0.78 SRC (0.41) CNR1HIF1ATSHRPDE4APDE4B
SCHEMBL5425818 0.77 ALDH1A2 (0.38) KDM4EALDH1A1
SCHEMBL27670851 0.75 POLB (0.33) CNR1POLBPDE4APDE4BPDE4C
SCHEMBL4516830 0.73 PDE4A (0.42) CNR1HIF1AMAT2ATSHRPDE4A
SCHEMBL4522660 0.73 CDK1 (0.39) CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1902201-A Bicyclic pyrimidin-4-(3H)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (VR1) MERCK SHARP & DOHME (GB) 2007-01-24 CN disclosed