SCHEMBL27672989

SCHEMBL27672989

O=C(Nc1ccsc1)c1ccc(CN2CCCCC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.62
HDAC1 Q13547 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
CYP2C9 P11712 3/20 0.56
KDM4E B2RXH2 2/20 0.56
ALDH1A1 P00352 2/20 0.56
HPGD P15428 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
ALOX15 P16050 1/20 0.56
RAB9A P51151 3/20 0.55
LMNA P02545 2/20 0.55
KMT2A Q03164 2/20 0.55
HTT P42858 2/20 0.55
GAA P10253 1/20 0.55
CYP3A4 P08684 1/20 0.54
HIF1A Q16665 3/20 0.53
EPAS1 Q99814 3/20 0.53
NPC1 O15118 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27652930 1.00 TNF (0.62) TNFHDAC1HDAC8HDAC6CYP2C9
SCHEMBL27672992 0.99 HDAC1 (0.61) TNFHDAC1HDAC8HDAC6CYP2C9
SCHEMBL27652919 0.96 HDAC6 (0.57) TNFHDAC1HDAC8HDAC6CYP2C9
SCHEMBL27672978 0.87 HIF1A (0.71) CYP2C9ALDH1A1CYP1A2CYP2D6ALOX15
SCHEMBL28759315 0.87 HDAC1 (0.53) TNFHDAC1HDAC6KDM4EALDH1A1
SCHEMBL27672993 0.86 RAB9A (0.66) TNFHDAC6KDM4EALDH1A1RAB9A
SCHEMBL27673031 0.86 NPC1 (0.54) RAB9AHIF1AEPAS1NPC1HRH3
SCHEMBL27672979 0.84 RAB9A (0.52) TNFHDAC6KDM4EALDH1A1RAB9A
SCHEMBL27652928 0.84 HIF1A (0.47) TNFHDAC6KDM4EALDH1A1RAB9A
SCHEMBL28663251 0.81 RAB9A (0.76) TNFHDAC1HDAC8HDAC6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1946395-A 1H-thieno [2, 3-c ] pyrazole derivatives useful as kinase inhibitors PHARMACIA ITALIA SPA (IT) 2007-04-11 CN claimed
CN-1946395-A 1H-thieno [2, 3-c ] pyrazole derivatives useful as kinase inhibitors PHARMACIA ITALIA SPA (IT) 2007-04-11 CN disclosed