SCHEMBL27675143

SCHEMBL27675143

Cc1c(NC(=O)n2cc(C(=O)O)c(=O)c3ccccc32)cccc1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 2/20 0.52
DHODH Q02127 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
S1PR1 P21453 4/20 0.42
S1PR3 Q99500 4/20 0.42
RBP4 P02753 4/20 0.41
CYP2C9 P11712 2/20 0.40
CFD P00746 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP3A4 P08684 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
LMNA P02545 1/20 0.40
CYP2D6 P10635 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
FABP4 P15090 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27693457 0.90 MEN1 (0.46) S1PR1S1PR3RBP4CYP2C9CYP2C19
SCHEMBL28766939 0.86 S1PR1 (0.43) S1PR1S1PR3RBP4CYP2C9CYP2C19
SCHEMBL27693502 0.84 KDM4E (0.44) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL27693589 0.80 S1PR1 (0.42) S1PR1S1PR3RBP4CYP2C9CYP2C19
SCHEMBL28768803 0.80 CNR2 (0.51) CYP2C9CYP2C19CYP3A4KDM4EALDH1A1
SCHEMBL27693559 0.79 KDM4E (0.51) CYP2C9CYP2C19CYP3A4KDM4EALDH1A1
SCHEMBL27675320 0.79 ALDH1A1 (0.46) S1PR1S1PR3KDM4EALDH1A1POLB
SCHEMBL27991300 0.78 KDM4E (0.43) CYP2C9CYP2C19CYP3A4KDM4EALDH1A1
SCHEMBL27693503 0.78 CFTR (0.47) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL27693495 0.78 LMNA (0.49) KDM4EALDH1A1POLBHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed