SCHEMBL27675155

SCHEMBL27675155

COc1ccc(-c2ccncc2CN)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
MGAT2 Q10469 1/20 0.43
PTGS2 P35354 5/20 0.43
PTGS1 P23219 2/20 0.43
KCNH2 Q12809 1/20 0.42
SLC6A2 P23975 4/20 0.41
SLC6A4 P31645 4/20 0.41
SLC6A3 Q01959 2/20 0.41
KMO O15229 1/20 0.39
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2E1 P05181 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2A6 P11509 2/20 0.39
CYP2B6 P20813 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP2C8 P10632 1/20 0.39
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12097845 0.76 CYP1A2 (0.46) MGAT2CYP1A2CYP2E1CYP2D6CYP2A6
SCHEMBL16841763 0.73 MEN1 (0.52) PTGS2PTGS1KMORAB9A
SCHEMBL31119316 0.72 CYP1A2 (0.51) MGAT2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL4483018 0.72 CYP1A2 (0.51) MGAT2SLC6A2SLC6A4SLC6A3CYP1A2
SCHEMBL12097501 0.72 LOXL2 (0.46) MGAT2CYP1A2CYP2E1CYP2D6CYP2A6
SCHEMBL6726046 0.72 PTGS2 (0.47) PTGS2PTGS1KCNH2RAB9A
SCHEMBL12097352 0.71 GPBAR1 (0.46) KCNH2
SCHEMBL12097552 0.71 LOXL2 (0.45) MGAT2CYP1A2CYP2E1CYP2D6CYP2A6
SCHEMBL12098015 0.70 LOXL2 (0.44) MGAT2SLC6A2SLC6A4SLC6A3CD274
SCHEMBL12326172 0.70 PTGS2 (0.53) ADORA2AADORA1PTGS2PTGS1KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1922144-A Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs MEMORY PHARM CORP (US) 2007-02-28 CN disclosed