SCHEMBL27675172

SCHEMBL27675172

CC(C)(C)OOC(=O)c1cccc(NCc2cncs2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HSD17B10 Q99714 2/20 0.44
TSHR P16473 1/20 0.44
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
EGFR P00533 1/20 0.41
KDR P35968 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
CTSL P07711 1/20 0.36
ABCB1 P08183 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.36
HIF1A Q16665 1/20 0.35
NAMPT P43490 1/20 0.35
HPGD P15428 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2908930 0.89 ABCB1 (0.44) TDP1ALDH1A1HSD17B10LMNAHTT
SCHEMBL27655242 0.86 TDP1 (0.44) TDP1ALDH1A1HSD17B10TSHRLMNA
SCHEMBL16160281 0.81 KMT2A (0.49) TDP1ALDH1A1HSD17B10TSHRLMNA
SCHEMBL26926495 0.80 AKR1C3 (0.51) TDP1LMNAHTTRAB9ANPC1
SCHEMBL27858128 0.75 PPARA (0.60) TDP1ALDH1A1HSD17B10TSHRLMNA
SCHEMBL2908569 0.74 NPC1 (0.43) TDP1LMNAHTTEGFRSMN1; SMN2
SCHEMBL224130 0.72 ALDH1A1 (0.75) TDP1ALDH1A1HSD17B10TSHRLMNA
SCHEMBL3451893 0.69 L3MBTL1 (0.57) ALDH1A1HSD17B10HTTEGFRRAB9A
SCHEMBL27960517 0.68 HIF1A (0.52) TDP1ALDH1A1HSD17B10TSHRLMNA
SCHEMBL5065687 0.68 TDP1 (0.68) TDP1ALDH1A1HSD17B10TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1922144-A Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs MEMORY PHARM CORP (US) 2007-02-28 CN disclosed