SCHEMBL27675219

SCHEMBL27675219

O=C(O)c1cn(C(=O)Nc2ccc(C(F)(F)F)cc2)c2ccccc2c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.48
CHRM1 P11229 1/20 0.47
NAMPT P43490 1/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
LMNA P02545 2/20 0.43
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43
TRPV1 Q8NER1 2/20 0.42
CREBBP Q92793 1/20 0.42
MCL1 Q07820 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
PTGS1 P23219 1/20 0.41
EPHX2 P34913 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
FAAH O00519 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28766934 0.88 CFTR (0.48) MAOBCHRM1LMNATRPV1EPHX2
SCHEMBL27675189 0.88 GRIK1 (0.51) RAB9ALMNACREBBPMAPTKMT2A
SCHEMBL27693487 0.88 LMNA (0.51) MAOBCHRM1LMNACREBBPSMN1; SMN2
SCHEMBL27675315 0.87 MEN1 (0.44) NAMPTRAB9ALMNASMN1; SMN2KDM4E
SCHEMBL27675384 0.87 CHRM1 (0.49) MAOBCHRM1LMNASMN1; SMN2KDM4E
SCHEMBL27693562 0.85 MAOB (0.51) MAOBCHRM1NAMPTTRPV1EPHX2
SCHEMBL27693550 0.85 NTRK1 (0.43) LMNAS1PR1S1PR3CREBBP
SCHEMBL27693544 0.85 CREBBP (0.42) CHRM1LMNAS1PR1S1PR3CREBBP
SCHEMBL28763086 0.84 CHRM1 (0.46) MAOBCHRM1LMNAS1PR1S1PR3
SCHEMBL28766931 0.84 CHRM1 (0.52) MAOBCHRM1NPC1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed