SCHEMBL27675231

SCHEMBL27675231

N#CCc1ccc(-c2ccccc2)c(N)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
HSD17B10 Q99714 2/20 0.48
MMP3 P08254 1/20 0.42
CSNK2A1 P68400 2/20 0.41
LMNA P02545 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
FLT3 P36888 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
ENPP2 Q13822 1/20 0.38
TNF P01375 1/20 0.37
KDM4E B2RXH2 2/20 0.36
HPGD P15428 1/20 0.36
DPP4 P27487 1/20 0.36
CYP19A1 P11511 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CG P48736 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5103341 0.81 MMP3 (0.44) MMP3CSNK2A1LMNAADORA2AADORA1
SCHEMBL29018975 0.81 MMP3 (0.44) ALDH1A1MMP3CSNK2A1LMNAFLT3
SCHEMBL396207 0.80 ALDH1A1 (0.54) ALDH1A1HSD17B10MMP3FLT3TNF
SCHEMBL12050457 0.79 ESR2 (0.49) ALDH1A1HSD17B10MMP3CSNK2A1LMNA
SCHEMBL17892098 0.79 CSNK2A1 (0.62) ALDH1A1HSD17B10MMP3CSNK2A1LMNA
Methane SCHEMBL7037141 0.79 MMP3 (0.42) MMP3CSNK2A1LMNAADORA2AADORA1
SCHEMBL3783312 0.78 CSNK2A1 (0.65) ALDH1A1HSD17B10CSNK2A1DPP4BACE1
SCHEMBL3786057 0.78 ALDH1A1 (0.50) ALDH1A1HSD17B10CSNK2A1BACE1
SCHEMBL28171242 0.77 ALDH1A1 (0.48) ALDH1A1HSD17B10CSNK2A1LMNABACE1
SCHEMBL13957118 0.77 CSNK2A1 (0.49) ALDH1A1HSD17B10CSNK2A1KDM4EDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891680-B Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-29 CN disclosed
CN-103641765-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2014-03-19 CN disclosed
CN-101935301-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2013-10-16 CN disclosed
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed