SCHEMBL27677406

SCHEMBL27677406

COC(=O)c1ccc(-c2ccc(Cl)cc2)s1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.63
KDM4E B2RXH2 4/20 0.56
NPC1 O15118 2/20 0.56
MAPT P10636 2/20 0.56
RAB9A P51151 2/20 0.56
CASP3 P42574 1/20 0.56
SENP8 Q96LD8 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
SENP6 Q9GZR1 1/20 0.56
ESRRG P62508 2/20 0.55
ESR1 P03372 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.51
ALDH1A1 P00352 3/20 0.51
HPGD P15428 2/20 0.51
GLA P06280 1/20 0.51
GAA P10253 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
CNR1 P21554 3/20 0.49
LMNA P02545 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6477476 0.91 KDM4E (0.58) IKBKBKDM4ENPC1MAPTRAB9A
SCHEMBL27141132 0.85 RAB9A (0.54) IKBKBKDM4ENPC1MAPTRAB9A
SCHEMBL497984 0.85 ESRRG (0.56) KDM4ENPC1MAPTRAB9AESRRG
SCHEMBL12348717 0.85 HSD17B1 (0.56) KDM4ENPC1MAPTRAB9AESRRG
SCHEMBL7259715 0.83 APP (0.53) IKBKBKDM4ENPC1MAPTRAB9A
SCHEMBL2491378 0.83 RAB9A (0.72) KDM4ENPC1MAPTRAB9AESRRG
SCHEMBL6805238 0.83 KDM4E (0.67) IKBKBKDM4ENPC1MAPTRAB9A
SCHEMBL2550687 0.83 KDM4E (0.72) KDM4ENPC1MAPTSMN1; SMN2ALDH1A1
SCHEMBL71536 0.83 RAB9A (0.66) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL1144728 0.83 IKBKB (0.58) IKBKBNPC1MAPTRAB9AESRRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100584840-C Substituted heterocyclic compounds and uses thereof ASTRAZENECA AB 2010-01-27 CN disclosed
CN-1922172-A Substituted heterocyclic compounds and uses thereof ASTRAZENECA AB (SE) 2007-02-28 CN disclosed